Aryl and hetaryl sulfonamides as active agents against abiotic plant stress 机翻标题: 暂无翻译,请尝试点击翻译按钮。

公开号/公开日
WO2011113861 A2 2011-09-22 [WO2011113861] WO2011113861 A3 2012-05-18 [WO2011113861] / 2011-09-22 2012-05-18
申请号/申请日
2011WO-EP53964 / 2011-03-16
发明人
FRACKENPOHL JENS; HEINEMANN INES; MUELLER THOMAS; VON KOSKULL-DOERING PASCAL; DITTGEN JAN; SCHMUTZLER DIRK; ROSINGER CHRISTOPHER HUGH; HAEUSER-HAHN ISOLDE; HILLS MARTIN JEFFREY
申请人
BAYER CROPSCIENCE
主分类号
IPC分类号
A01N-043/08;A01N-043/12;A01N-043/36;A01N-043/38;A01N-043/40;A01N-043/42;A01N-043/56;A01N-043/72;A01N-043/78;A01N-043/80;A01P-021/00
摘要
(WO2011113861)
The invention relates to the use of substituted sulfonamides of the general formula (I), or the salts thereof, for boosting the stress tolerance in plants to abiotic stress, in particular for boosting the plant growth and/or increasing the plant yield.
机翻摘要
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地址
代理人
代理机构
优先权号
2010EP-0156922 2010-03-18 2010US-61315583 2010-03-19
主权利要求
(WO2011113861)
1. Use of substituted substituted sulfonamides of the formula (I) or their salts to increase tolerance to abiotic stress in plants, wherein A (1), A (2), A (3) are the same or different and independently of each other, N (nitrogen) or the group CW are, however, more than two N atoms are adjacent in any case, and wherein W the grouping CW are identical or different meanings as defined below, has W are each hydrogen, nitro, amino, cyano, thiocyanato, Isothiocyanato, halogen, alkyl, cycloalkyl, alkenyl, alkynyl, aryl, arylalkyl, arylalkoxy, heteroaryl, alkoxyalkyl, haloalkyl, halocycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, hydroxycarbonyl, aminocarbonyl, alkylaminocarbonyl, cycloalkylaminocarbonyl, alkylamino, alkylthio, haloalkylthio, Bisalkylamino, cycloalkylamino, alkylcarbonylamino Cycloalkylcarbonylamino, formylamino, Haloalkylcarbonylamino, alkoxycarbonylamino, (alkyl) aminocarbonylamino, alkylsulfonylamino, Cycloalkylsulfonylamino, arylsulfonylamino, Hetarylsulfonylamino, Sulfonylhaloalkylamino, Aminoalkylsulfonyl, Aminohaloalkylsulfonyl, alkylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, alkylsulfinyl, Cycloalkylsulfinyl, arylsulfinyl, N, S-Dialkylsulfonimidoyl, S Alkylsulfonimidoyl, alkylsulphonylaminocarbonyl, Cycloalkylsulfonylaminocarbonyl, Cycloalkylaminosulfonyl R (1) is H, nitro, amino, cyano, halogen, alkyl, cycloalkyl, alkenyl, alkynyl, Aryl, arylalkyl, heteroaryl, alkoxyalkyl, haloalkyl, halocycloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkoxycarbonyl, Hydroxy, aminocarbonyl, Alkylaminocarbonyl, alkylamino, Bisalkylamino, Cycloalkylamino, Alkylcarbonylamino, Cycloalkylcarbonylamino, formylamino, Haloalkylcarbonylamino, Alkoxycarbonylamino, (alkyl) aminocarbonylamino, sulphonylamino, alkylsulphonylamino, Haloalkylsulfonylamino, Cycloalkylsulfonylamino, Aminoalkylsulfonyl, Aminohaloalkylsulfonyl, alkylsulfonyl, Cycloalkylsulfonyl, arylsulfonyl, Alkylsulfinyl, Cycloalkylsulfinyl, Arylsulfinyl, N, S-Dialkylsulfonimidoyl, S Alkylsulfonimidoyl, Alkylsulphonylaminocarbonyl, Cycloalkylsulfonylaminocarbonyl, Cycloalkylaminosulfonyl is, R (2) is H, nitro, amino, cyano, halogen, alkyl, cycloalkyl, alkenyl, alkynyl, aryl, arylalkyl, heteroaryl, alkoxyalkyl, haloalkyl, halocycloalkyl, Alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkoxycarbonyl, Hydroxy, aminocarbonyl, Alkylaminocarbonyl, alkylamino, Bisalkylamino, Cycloalkylamino, Alkylcarbonylamino, Cycloalkylcarbonylamino, formylamino, Haloalkylcarbonylamino, Alkoxycarbonylamino, (alkyl) aminocarbonylamino, sulphonylamino, Alkylsulphonylamino, Haloalkylsulfonylamino, Cycloalkylsulfonylamino, Aminoalkylsulfonyl, Aminohaloalkylsulfonyl, alkylsulfonyl, Cycloalkylsulfonyl, arylsulfonyl, Alkylsulfinyl, Cycloalkylsulfinyl, Arylsulfinyl, N, S-Dialkylsulfonimidoyl, S Alkylsulfonimidoyl, Alkylsulphonylaminocarbonyl, Cycloalkylsulfonylaminocarbonyl, Cycloalkylaminosulfonyl, R (1) and R (2) with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated, optionally interrupted by hetero atoms and optionally further substituted 5 to 7-membered ring, R (1) and A (3), when A (3) is a group CW, with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated, optionally interrupted by hetero atoms and optionally further substituted 5 to 7 - membered ring, X is H, alkyl, alkylalkenyl, alkynyl, alkylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, heteroarylcarbonyl, alkoxycarbonyl, alkylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, Alkoxycarbonylcarbonyl, Arylalkoxycarbonylcarbonyl, alkylaminothiocarbonyl, Alkylaminocarbonyl, arylalkyl, Hetaroarylalkyl, cyanoalkyl, haloalkyl, cycloalkyl, cycloalkylalkyl, Y alkandiyl, cycloalkanediyl Alkenediyl, alkinediyl, Alkylalkendiyl, Arylalkandiyl, Alkoxydiyl, Alkoxyalkyldiyl, Alkylthioalkyldiyl, AI kylsulfinylal kyldiyl, Alkylsulfonylalkyldiyl or a direct bond between N and Q, Q is a phenyl ring or a 5 -, 6 - or 7-membered saturated or unsaturated heterocyclic ring or a 9 - or 10 - membered-fused bicyclic or tricyclic ring system, which optionally contains further hetero atoms, wherein the respective aforementioned ring or ring system optionally is mono-or polysubstituted by identical or different substituents, and wherein the substituents are independently selected from H, halogen, cyano, nitro, branched or unbranched alkyl, cycloalkyl, alkoxycycloalkyl, arylcycloalkyl, cycloalkyl, cycloalkyl, cycloalkylalkyl, alkenyl, alkynyl, arylalkyl, alkoxyalkyl, haloalkyl, halocycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, hydroxycarbonyl, aminocarbonyl, alkylaminocarbonyl, amino, alkylamino, Bisalkylamino, cycloalkylamino, alkylcarbonylamino, alkylcarbonyl, alkylthio, Haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl or the Substituents are independently selected from phenyl or a 5 - or 6-membered heteroaromatic ring, said phenyl or heteroaromatic ring being optionally mono-or polysubstituted by identical or different alkyl, alkenyl, alkynyl, cycloalkyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halogen, cyano, nitro, alkoxy, haloalkoxy, alkylthio, haloalkylthio substituted.
2.
2. Use according to claim 1, wherein in formula (I) A (1), A (2), A (3) are the same or different and independently of each other, N (nitrogen) or the group CW are, however, more than two N atoms are adjacent in any case, and wherein W the grouping CW may each have identical or different meanings as defined below; W are each hydrogen, nitro, amino, cyano, halogen, (d-C6)-alkyl, (C
-C
) cycloalkyl, (C
,-C
) alkenyl, ( C
, C
) alkynyl, aryl, aryl-(CrC
) - alkyl, heteroaryl, (Ci-C
) alkoxy (Ci-C
)-alkyl, (Ci-C
)-haloalkyl, (C
, C
)-halocycloalkyl, (Ci-C
) alkoxy, aryl (Ci-C
) alkoxy, ( Ci-C
) - haloalkoxy, (d-C 6)-alkoxycarbonyl, hydroxy, aminocarbonyl, (CRC6)-alkyl aminocarbonyl, (C 3-C
) cycloalkylaminocarbonyl, (Ci-Ce) - alkylamino, (C- C.
)-alkylthio, (Ci-C
)-haloalkylthio, bis-(Ci-C
) - alkylamino, (C3-C
)-cycloalkylamino, (CRC6)-alkylcarbonylamino, ( C3-C
) Cycloalkylcarbonylamino, formylamino, (Ci-Ce) - Haloalkylcarbonylamino, (CRC6) Alkoxycarbonylamino, (Ci-Ce) - (alkyl) aminocarbonylamino, (Ci-C6) alkylsulphonylamino, (C 3-C
) - Cycloalkylsulfonylamino, Arylsulfonylamino, Hetarylsulfonylamino, sulfonyl (Ci-C6) haloalkylamino, amino, (Ci-C6) alkylsulfonyl, amino (Ci-C
)-haloalkylsulfonyl, (Ci-C
) alkylsulfonyl, (C
, C
) - cycloalkylsulfonyl, arylsulfonyl, (Ci-C
)-Al kylsulfinyl, (C
-C
) - Cycloalkylsulfinyl, Arylsulfinyl, N, S-di-(Ci-C6) alkylsulfonimidoyl, S-(Ci-C6) Alkylsulfonimidoyl-, (Ci-C6) alkylsulfonylaminocarbonyl, (C3-C8) Cycloalkylsulfonylaminocarbonyl, (Ci-C6)-Cycloalkylaminosulfonyl, represents H, nitro, amino, cyano, halogen, (Ci-C 6)-alkyl, (C3 -C8)-cycloalkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl, aryl (Ci-C
) alkyl, heteroaryl,, (Ci-C
)-Al koxy-(Ci-C
)-alkyl, (CrC
) Haloal alkyl, (C
, C
) Halocycloal alkyl, (CrC
) alkoxy, (Ci-C
)-haloalkoxy, (Ci-C
)-alkylthio, (Ci-C
) - haloalkylthio, (Ci-C6)-alkoxycarbonyl, hydroxy, Aminocarbonyl, (Ci-C6)-alkyl aminocarbonyl, (C3-C8) - cycloalkylaminocarbonyl, (CRC6)-alkylamino, bis (CRC6)-alkylamino, (C3-C8)-Cycloalkylamino, (Ci-C6) Alkylcarbonylamino, (C3 -C8) - Cycloalkylcarbonylamino, formylamino, (C1-C6) - Haloalkylcarbonylamino, (Ci-C6) Alkoxycarbonylamino, (d-C6) - (alkyl) aminocarbonylamino, (Ci-C6) alkylsulphonylamino, (C3-C8) - Cycloalkylsulfonylamino, arylsulfonylamino, Hetarylsulfonylamino, sulfonyl (Ci-C6)-haloalkylamino, amino (Ci-C6) alkylsulfonyl, amino, (CrC
)-haloalkylsulfonyl, (Ci-C
) alkylsulfonyl, (C [ 3], C
) - cycloalkylsulfonyl, arylsulfonyl, (C 1-C
)-alkyl below If i nyl, (C
, C
) - cycloalkyl kylsulfinyl, arylsulfinyl, N, S -di-(Ci-C6) alkylsulfonimidoyl, S-(CRC6) Alkylsulfonimidoyl, (CRC6) alkylsulphonylaminocarbonyl, (C3-C8) Cycloalkylsulfonylaminocarbonyl, (Ci-C6) Cycloalkylaminosulfonyl stands for H, nitro, amino, cyano, halogen, (Ci-C6)-alkyl, (C3-C8) cycloalkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl, aryl- (Ci-C
) alkyl, heteroaryl, (Ci-C
)-Al koxy-(Ci-C
)-alkyl, (Ci-C
) Haloal alkyl, ( C
, C
) Halocycloal alkyl, (Ci-C
) alkoxy, (Ci-C
)-haloalkoxy, (Ci-C
)-alkylthio, (Ci- C
) - Haloalkylthio, (d-C 6)-alkoxycarbonyl, hydroxy, Aminocarbonyl, (Ci-C6)-alkyl aminocarbonyl, (C3-C8) - cycloalkylaminocarbonyl, (Ci-C6) alkylamino, bis-(Ci-C 6)-alkylamino, (C3-C8)-Cycloalkylamino, (Ci-C6) - Alkylcarbonylamino, (C3-C8) - Cycloalkylcarbonylamino, formylamino, (C 1-C 6) - Haloalkylcarbonylamino, (Ci-C6) Alkoxycarbonylamino, (d-C6) - (alkyl) aminocarbonylamino, (Ci-C6) alkylsulphonylamino, (C3-C8) - Cycloalkylsulfonylamino, Arylsulfonylamino, Hetarylsulfonylamino, sulfonyl (Ci-C6) - aloalkylamino, amino-(Ci-C 6)-alkylsulfonyl, amino (Ci-C
)-haloalkylsulfonyl, (Ci-C
) alkylsulfonyl, (C
, C
) - cycloalkylsulfonyl, arylsulfonyl, (C1-C
) - AI ky I su If i ny I, (C
-C
) - Cycloalkylsulfinyl, Arylsulfinyl, N, S-di-(Ci-C6) alkylsulfonimidoyl, S-(Ci-C6) Alkylsulfonimidoyl, (CRC6) - alkylsulphonylaminocarbonyl, (C3-C8) - Cycloalkylsulfonylaminocarbonyl, (Ci-C6) Cycloalkylaminosulfonyl is, R (1) and R (2), with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated, optionally interrupted by hetero atoms and optionally further substituted 5 to 7-membered ring, R (1) and A (3), when A (3) is a group CW, with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated, optionally interrupted by hetero atoms and optionally further substituted 5 to 7 - membered ring, X is H, (Ci-C
)-alkyl, (Ci-C
) alkyl (C2-C
) alkenyl, (Ci-C
) - alkylcarbonyl, (C3 -C8)-Cycloalkylcarbonyl, aryl carbonyl, Heteroarylcarbonyl, (d-C 6)-alkoxycarbonyl, (CRC6) alkylsulfonyl, (C
-C
) cycloalkylsulfonyl, arylsulfonyl, (d-Ce) - Alkoxycarbonylcarbonyl, aryl (Ci-C6) alkoxycarbonylcarbonyl, (C1-C6) - alkylaminothiocarbonyl, (Ci-C6)-alkylaminocarbonyl, aryl-(Ci-C6) alkyl, heteroaryl (Ci-C
) alkyl, (C
, C
) -alkynyl, (Ci-C
)-cyanoalkyl, (Ci-C
) - haloalkyl, (C
, C
) cycloalkyl, (C
, C
) -cycloalkyl-(Ci-C
) alkyl is (Ci-C
)-alkanediyl, (C
, C
) alkynyl, (C
, C
)-cycloalkanediyl or (C
, C
) - Al kendiyl, (C1-C
)-alkyl-(C
, C
) al kendiyl, aryl-(C -C
) al kandiyl, (C1-C
)-Al koxydiyl, (C1-C
)-Al koxy-(Ci-C
) kyldiyl al, (C1-C
) - alkoxycarbonyl, (Ci- C.
) alkyldiyl, (C1-C
)-Al kylth io-(Ci-C
) kyldiyl al, (C1-C
)-Al kylsulfinyl-(Ci-C [ 6]) kyldiyl al, (Ci-C
) alkylsulfonyl, (Ci-C
) - al kyldiyl or a direct bond between N and Q stands for a phenyl ring or a 5 -, 6 -, or 7-membered saturated or unsaturated heterocyclic ring or a 9 - or 10-membered-fused bicyclic or tricyclic ring system, which may contain further hetero atoms, if appropriate, the respective above-mentioned ring or ring system is optionally mono-or polysubstituted by identical or different substituents, and wherein the substituents are independently selected from H, halogen, cyano, nitro, branched or unbranched (C1-C-6) - Alkyl, (C
, C
) cycloalkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl (Ci-C
) - alkyl, (Ci-C
) alkoxy (Ci-C
)-alkyl, (Ci-C
)-haloalkyl, (C
, C
) - Halocycloal alkyl, (C
-C
)-Al koxycycloal alkyl, (C
-C
) Arylcycloal alkyl, (C
-C
)-cycloalkyl alkyl-(C
-C
)-cycloalkyl alkyl, (C
-C
)-cycloalkyl alkyl-(Ci-C [ 6])-alkyl, (Ci-C
) alkoxy, (Ci-C
)-haloalkoxy, (Ci-C
) alkoxycarbonyl, Hydroxycarbonyl, aminocarbonyl, (CRC6)-alkylaminocarbonyl, amino, (CRC6)-alkylamino, bis-(Ci-C6)-alkylamino, (C
, C
)-cycloalkylamino, (Ci-C
) -alkylcarbonylamino, (Ci-C
) alkylcarbonyl, (Ci-C
)-alkylthio, (Ci-C
)-haloalkylthio, (C1-C
) Haloal kylsulfinyl, (C -C
) - haloalkylsulfonyl, or wherein the substituents are independently selected from phenyl or a 5 - or 6-membered heteroaromatic ring, said phenyl or heteroaromatic ring being optionally mono-or polysubstituted, identically or differently, with (d-C6) alkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, (C
, C
) cycloalkyl, (Ci-C
)-haloalkyl, (C
, C
) Haloal kenyl, (C
, C
) Haloal alkynyl, (C
, C
) Halocycloal alkyl, halogen, cyano, nitro, (Ci-C
) alkoxy, (Ci-C
)-haloalkoxy, (Ci-C
) - are alkylthio, (Ci-C
)-haloalkylthio substituted and Q furthermore represents one of the radicals Q-1 to Q-192 Q 1 Q 2 Q 3 Q 4 Q 5 Q-6 I Br Q-9 Q-20 Q-2 Q-22 Q-23 Q-24 he F ^ Cl Q-31 Q-32 Q-33 Q-34 Q-35 Q-36 Q-37 Q-38 Q-39 Q-40 Q-41 Q-42 F N NT N FF Q-43 Q-44 Q-45 Q-46 Q-47 Q-48.
3.
3. Ί3 3CO 3 35 ^ 0 3\\Q-73 Q-74 Q-75 Q-76 Q-77 Q-78ΝΗΗ ΗQ-91 Q-92 Q-93 Q-94 Q-95 Q-96 HH \\Q-97 Q-98 Q-99 Q-100 Q-101 Q-102Q-151 Q-152 Q-153 Q-154 Q-155 Q-156ΝQ-157 Q-158 Q-159 Q-160 Q-161 Q-162
3.
3. Use according to claim 2, wherein in formula (I) A (1), A (2), A (3) are the same or different and independently of each other, N (nitrogen) or the group CW are, however, more than two N atoms are adjacent in any case, and wherein W the grouping CW each has identical or different meanings as defined below; W are each hydrogen, nitro, amino, cyano, halogen, (DC
) alkyl, (C
C.
) cycloalkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl, aryl-(dC
) - alkyl, heteroaryl, (Ci-C
) alkoxy (Ci-C
) alkyl (DC
)-haloalkyl, (C
, C
)-halocycloalkyl, (CC
) alkoxy, aryl (Ci-C
) alkoxy, (DC [4 ]) - haloalkoxy, (dC
)-alkoxycarbonyl, hydroxy, aminocarbonyl, (CrC
)-alkyl aminocarbonyl, (C 3-C
) cycloalkylaminocarbonyl, (Ci-C
) - alkylamino, ( dC
) alkylthio, (Ci-C
) Haloalkylthio, bis-(dC
) - alkylamino, (C3-C6) Cycloalkylamino, (Ci-C
) Alkylcarbonylamino, ( C3-C
) Cycloalkylcarbonylannino, formylamino, (Ci-C
) - Haloalkylcarbonylamino, (Ci-C
) Alkoxycarbonylamino, (Ci-C
) - (alkyl) Aminocarbonylannino, ( Ci-C
) alkylsulfonylamino, (C3-C6) - Cycloalkylsulfonylamino, arylsulfonylamino, Hetarylsulfonylamino, sulfonyl (Ci-C
)-haloalkylamino, amino (Ci-C
) alkylsulfonyl, amino, (Ci-C
) haloalkylsulfonyl, (Ci-C
)-alkylsulfonyl, (C 3-C
) - cycloalkylsulfonyl, arylsulfonyl, (Ci-C
) Alkylsulfinyl, (C [3 ]-C
) - Cycloalkylsulfinyl, arylsulfinyl, N, S-di-(Ci-C
) alkylsulfoninnidoyl, S-(Ci-C
) Alkylsulfonimidoyl, (Ci-C
) -alkylsulphonylaminocarbonyl, (C3-C
) - Cycloalkylsulfonylaminocarbonyl, (Ci-C
) is Cycloalkylaminosulfonyl, H, nitro, amino, cyano, halogen, (Ci-C
) alkyl, (C
C.
) cycloalkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl, aryl (Ci-C [4 ]) alkyl, heteroaryl, (Ci-C
) alkoxy-(C
to C
) alkyl, (CrC
)-haloalkyl, (C
, C
)-halocycloalkyl, (dC
) alkoxy, (DC
)-haloalkoxy, (DC
)-alkylthio, (dC)
- haloalkylthio, (DC
) alkoxycarbonyl, hydroxycarbonyl, Aminocarbonyl, (Ci-C
)-alkylaminocarbonyl, (C3-C
) - cycloalkylaminocarbonyl, (CrC
)-alkylamino, bis-(Ci-C
)-alkylamino, (C
-C 6)-Cycloalkylamino, (Ci-C
) Alkylcarbonylamino, (C 3-C
) - Cycloalkylcarbonylamino, formylamino, (Ci-C
) - Haloalkylcarbonylamino, (CrC [4 ]) Alkoxycarbonylamino, (dC
) - (alkyl) aminocarbonylamino, (Ci-C
) alkylsulphonylamino, (C3-C6) - Cycloalkylsulfonylamino, Arylsulfonylamino, Hetarylsulfonylamino, Sulfonyl (Ci-C
)-haloalkylamino, amino (Ci-C
) alkylsulfonyl, amino (Ci-C
)-haloalkylsulfonyl, (Ci-C
) alkylsulfonyl, ( C3-C
) - cycloalkylsulfonyl, arylsulfonyl, (C 1-C
)-alkyl below If i nyl, (C
, C
) - Cycloalkylsulfinyl, arylsulfinyl, N, S-di - (Ci-C
) alkylsulfonimidoyl, S-(Ci-C
) Alkylsulfonimidoyl, (Ci-C) alkylsulfonylaminocarbonyl, (C
, C
) - Cycloalkylsulfonylaminocarbonyl, (Ci-C
) Cycloalkylaminosulfonyl, R (2) is H, nitro, amino, cyano, halogen, (DC
) alkyl, (C
, C
) - cycloalkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl, aryl-(CrC
) alkyl, heteroaryl, (Ci-C [ 4])-Al koxy-(Ci-C
)-alkyl, (Ci-C
) Haloal alkyl, (C
, C
) Halocycloal alkyl, (Ci-C
) alkoxy, (DC
)-haloalkoxy, (Ci-C
)-alkylthio, (dC)
- haloalkylthio, (Ci-C
) alkoxycarbonyl, hydroxycarbonyl, Aminocarbonyl, (Ci-C
)-alkylaminocarbonyl, (C3-C
) - cycloalkylaminocarbonyl, (CrC
)-alkylamino, bis-(Ci-C
)-alkylamino, (C3-C6 ) Cycloalkylamino, (Ci-C
) Alkylcarbonylamino, (C3-C7) - Cycloalkylcarbonylamino, formylamino, (Ci-C
) - Haloalkylcarbonylamino, (Ci-C
) Alkoxycarbonylamino, (dC [ 4]) - (alkyl) aminocarbonylamino, (Ci-C
) alkylsulfonylamino, (C3-C6) - Cycloalkylsulfonylamino, arylsulfonylamino, Hetarylsulfonylamino, sulfonyl (Ci-C
)-haloalkylamino, amino-(Ci- C
) alkylsulfonyl, amino (Ci-C
)-haloalkylsulfonyl, (CrC
) alkylsulfonyl, (C3-C
) - cycloalkylsulfonyl, arylsulfonyl, (C 1-C [4 ]) - AI kyl su If i ny I, (C 3-C
) - Cycloalkylsulfinyl, Arylsulfinyl, N, S-di-(Ci-C
) alkylsulfonimidoyl, S-(Ci-C
) Alkylsulfonimidoyl, (Ci-C
) alkylsulphonylaminocarbonyl, (C3-C7) - Cycloalkylsulfonylaminocarbonyl, (CrC
) Cycloalkylaminosulfonyl is, R (1) and R (2), with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated, optionally interrupted by hetero atoms and optionally further substituted 5 or 6-membered ring, R (1) and A (3), when A (3) is a group CW, with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated, optionally interrupted by hetero atoms and optionally further substituted 5 to 6 - membered ring, is H, (Ci-C
) alkyl, (Ci-C
) alkyl-(C
, C
) alkenyl, (Ci-C [ 4]) - alkylcarbonyl, (C3-C6) Cycloalkylcarbonyl, aryl carbonyl, Heteroarylcarbonyl, (Ci-C
) Al-alkoxycarbonyl, (Ci-C
) Al kylsulfonyl, (C3-C6) cycloalkylsulfonyl, arylsulfonyl, (DC
) alkoxycarbonyl-carbonyl, aryl-(CrC
) alkoxycarbonylcarbonyl, (Ci-C
) - alkylaminothiocarbonyl, (Ci-C
)-alkylaminocarbonyl, aryl-(CRC4) alkyl Hetaroaryl-(Ci-C
) alkyl, (C
, C
) alkynyl, (Ci-C
) cyanoalkyl, (dC)
- haloalkyl, (C
, C
) cycloalkyl, (C
, C
) cycloalkyl (Ci-C
)-alkyl, for (Ci-C
)-alkanediyl, (C
, C
)-cycloalkanediyl or (C
, C
)-alkenediyl, (C
, C
) - alkynediyl, (Ci-C
) alkyl-(C
, C
)-alkenediyl, aryl (dC
)-alkanediyl, (CC
) - Al koxyd iyl, (C 1-C
) - AI alkoxy-(C 1-C
) al kyld iyl, (Ci-C
) Al-alkoxycarbonyl - (Ci-C
) al kyldiyl, (Ci-C
) Al-alkylthio-(d-C
) al kyldiyl, (Ci-C
) - Al kylsulfinyl-(Ci-C
) al kyldiyl, ( Ci-C
)-alkylsulfonyl (Ci-C
) alkyldiyl or a direct bond between N and Q stands for a phenyl ring or a 5 -, 6 - or 7-membered saturated or unsaturated heterocyclic ring or 9 - or 10-membered-fused bicyclic or tricyclic ring system, which optionally contains further hetero atoms, wherein the respective aforementioned ring or ring system is optionally mono-or polysubstituted by identical or different substituents, and wherein the substituents are independently selected from H, Halogen, cyano, nitro, branched or unbranched (dC
) alkyl, (C
, C
) cycloalkyl-alkyl, (C
, C
)-Al koxycycloal alkyl, ( C
-C
) Arylcycloal alkyl, (C
-C
)-cycloalkyl alkyl-(C
-C
)-cycloalkyl alkyl, (C
- C.
) alkyl-cycloalkyl-(Ci-C
)-alkyl, (C
, C
) alkenyl, (C
, C
) alkynyl, aryl, - (dC
) alkyl, (DC
) alkoxy (dC
) alkyl, (Ci-C
)-haloalkyl, (C
, C
) -halocycloalkyl, (DC
) alkoxy, (CrC
)-haloalkoxy, (DC
) alkoxycarbonyl, hydroxycarbonyl, Aminocarbonyl, (CrC
)-alkylaminocarbonyl, amino, (CrC
) - alkylamino, bis-(CrC
)-alkylamino, (C
-C6)-cycloalkylamino, (Ci-C [4 ]) - alkylcarbonylamino, (Ci-C
) alkylcarbonyl, (Ci-C
)-alkylthio, (C1-C4) - haloalkylthio, (Ci-C)-haloalkylsulfinyl, (CRC)-haloalkylsulfonyl, or wherein the substituents are independently selected from phenyl or a 5 - or 6-membered heteroaromatic ring, said phenyl or heteroaromatic ring being optionally mono-or polysubstituted by identical or different (Ci-C
) alkyl, (C-2-C6 ) alkenyl, (C
, C
) alkynyl, (C
, C
) cycloalkyl, (Ci-C
)-haloalkyl, (C
-C
) - haloalkenyl, (C2-C6)-haloalkynyl, (C3-C6) halocycloalkyl, halogen, cyano, nitro, (dC
)-alkoxy, (Ci-C
)-haloalkoxy, ( Ci-C
)-alkylthio, (dC)
-haloalkylthio further substituted, and Q represents one of the above-described radicals Q-1 to Q-192.
4.
4. Use according to claim 2, wherein in formula (I) A (1), A (2), A (3) are the same or different and independently of each other, N (nitrogen) or the group CW are, however, more than two N atoms are adjacent in any case, and wherein W the grouping CW each has identical or different meanings as defined below; W are each hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, (DC
) alkoxy, (Ci-C
) alkyl, (C
, C
) -alkenyl, cyclopropyl, cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, methylamino, trifluoromethyl, Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (1) is hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, (Ci-C
) - alkoxy, (Ci-C
) alkyl, (C
-C
) alkenyl, cyclopropyl, cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, (Ci-C
) alkylamino, trifluoromethyl; Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (2) is hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, (Ci-C 4)-alkyl, (C2-C6)-alkenyl, cyclopropyl, Cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, (CrC
) alkylamino, trifluoromethyl; Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (1) and R (2), with the atoms to which they are attached form a fully saturated or fully unsaturated 5 - to 6-membered carbocyclic or heterocyclic ring, which is optionally further substituted by nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, methyl, ethyl, cyclopropyl, Methylcarbonylamino, methylamino, trifluoromethyl, trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, Methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, R (1) and A (3), when A (3) is a group CW, with the atoms to which they are attached form a fully saturated or fully unsaturated 5 - to 6-membered carbocyclic or heterocyclic ring, is optionally further substituted by nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, methyl, ethyl, cyclopropyl, methylcarbonylamino, methylamino, trifluoromethyl, trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl dimethylamino, benzyloxy, phenyl, H, methyl, ethyl, n-propyl, cyclopropyl, isopropyl, methylcarbonyl, ethylcarbonyl, 2'-trifluoromethyl-4'-pyridylcarbonyl, cyclopropyl, benzyl, CH
-pyridyl, N- propylcarbonyl, tert-butylcarbonyl, Cyclobutylcarbonyl, cyclopentylcarbonyl, cyclohexyl-, Methoxycarbonyl, ethoxycarbonyl, allyl, ethynyl, prop-1-in-3-yl, but-2-in-3-yl, cyanomethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2,2,3, 3.3 - pentafluoropropyl, 3,3,2,2-tetrafluoropropyl, 4,4,4-trifluorobutyl, Methoxycarbonylmethyl stands for CH
, CH
CH
, CH (CH
), CH (CO
Me) CH
, CH (CF
), spiro-cyclo propylene, represents an optionally singly or multiply substituted Phenyl or an unsubstituted or mono-or polysubstituted substituted 5 -, 6 - or 7-membered saturated or unsaturated heterocyclic ring or a 9 - or 10-membered-fused heterobicyclic ring system of the above-described series of Q-1 is-Q-192, where the substituents are independently selected from hydrogen, methyl, ethyl, n-propyl, iso-propyl, cyclopropyl, methyl-cyclopropyl, methoxy, ethoxy, trifluoromethyl, fluorine, chlorine, bromine, iodine, cyano, nitro, trifluoromethoxy, methylthio, trifluoromethylthio, OCHF
OCCIF
, methoxycarbonyl, phenyl, p-chlorophenyl, m-chlorophenyl, o-chlorophenyl, ο, ρ-dichlorophenyl, m, m-dichlorophenyl, o-iodophenyl, m-iodophenyl, p-iodophenyl, o-bromophenyl, m-bromophenyl, p -bromophenyl, o-methylphenyl, m-methylphenyl, p-methylphenyl, o-fluorophenyl, m-fluorophenyl, p-fluorophenyl, o-methoxyphenyl, m-methoxyphenyl, p-methoxyphenyl, o-Thfluormethylphenyl, m Thfluornnethylphenyl, p-trifluoromethylphenyl, p-trifluoromethoxyphenyl, p-trifluoromethylthiophenyl, o-nitrophenyl, m-nitrophenyl, p-nitrophenyl, o-cyanophenyl, m-cyanophenyl, p-cyanophenyl.
5.
5. Use according to claim 2, wherein in formula (I) A (1), A (2), A (3) are the same or different and independently of each other, N (nitrogen) or the group CW are, however, more than two N atoms are adjacent in any case, and wherein W the grouping CW are identical or different meanings as defined below, has W are each hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, (CrC
) alkoxy, (DC
) alkyl, (C
,-C
) alkenyl, cyclopropyl, cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, methylamino, trifluoromethyl, Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonyl, methyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (1) is hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, (C1-C4) - alkoxy, (DC
) alkyl, (C
, C
) - alkenyl, cyclopropyl, cyclobutyl, Methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, (CrC
) alkylamino, trifluoromethyl; Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is R (2) is hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, (Ci-C
) alkyl, (C2-C6)-alkenyl, cyclopropyl, Cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, (CRC4)-alkylamino, trifluoromethyl, Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (1) and R (2), with the atoms to which they are attached form a fully saturated or fully unsaturated 5 - to 6-membered carbocyclic or heterocyclic ring, which is optionally further substituted by nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, methyl, ethyl, cyclopropyl, Methylcarbonylamino, methylamino, trifluoromethyl, trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, Methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, R (1) and A (3), when A (3) is a group CW, with the atoms to which they are attached form a fully saturated or fully unsaturated 5 - to 6-membered carbocyclic or heterocyclic ring, which is optionally further substituted by nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, methyl, ethyl, cyclopropyl, methylcarbonylamino, methylamino trifluoromethyl, trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, Phenyl, X is H, methyl, ethyl, n-propyl, cyclopropyl, isopropyl, methylcarbonyl, ethylcarbonyl, 2'-trifluoromethyl-4'-pyridylcarbonyl, Cydopropylcarbonyl, benzyl, CH-pyridyl, n-propylcarbonyl, tert-butylcarbonyl, cyclobutylcarbonyl, cyclopentylcarbonyl, cyclohexyl-, Methoxycarbonyl, ethoxycarbonyl, allyl, ethynyl, prop-1-in-3-yl, but-2-in-3-yl, cyanomethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2,2,3, 3.3 - pentafluoropropyl, 3,3,2,2-tetrafluoropropyl, 4,4,4-trifluorobutyl, Methoxycarbonyl methyl; Y is CH
, CH
CH
, CH (CH
), CH (CO
Me) CH
, CH (CF
), spiro-cyclo propylene is, Q is a moiety selected from the above series Q-2 is to Q-192.
6.
6. Use according to claim 2, wherein in formula (I) A (1), A (2), A (3) are the same or different and independently of each other, N (nitrogen) or the group CW are, however, more than two N atoms are adjacent in any case, and wherein W the grouping CW are identical or different meanings as defined below, has W are each hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, (DC
) alkoxy, (DC
) alkyl, (C
,-C
) alkenyl, cyclopropyl, cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, methylamino, trifluoromethyl, Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl, R (1) is hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, (Ci-C
) - alkoxy, (Ci-C
) alkyl, (C [2 ] C.
) alkenyl, cyclopropyl, cyclobutyl, Methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, (CRC4)-alkylamino, trifluoromethyl, Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (2) is hydrogen, nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, (DC
) alkyl, (C
, C
) alkenyl, cyclopropyl, cyclobutyl, methylcarbonylamino, Cyclopropylcarbonylamino, Cyclobutylcarbonylamino, (Ci-C
) alkylamino, trifluoromethyl; Trifluoromethylthio, trifluoromethoxy, difluoromethoxy, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, dimethylamino, benzyloxy, phenyl, Methylsulfonylaminocarbonyl, Cyclopropylsulfonylaminocarbonyl, cyclopropylaminocarbonyl, Cyclopropylaminosulfonyl is, R (1) and R (2), with the atoms to which they are attached form a fully saturated or fully unsaturated 5 - to 6-membered carbocyclic or heterocyclic ring, which is optionally further substituted by nitro, amino, cyano, fluorine, chlorine, bromine, iodine, methoxy, ethoxy, isopropoxy, methyl, ethyl, cyclopropyl, (...)
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