COMPOSITES HETEROCICLICOS, INSECTICIDAL PROCESS FOR ITS PREPARACAO, COMPOSICOES, PROCESS FOR COMBAT the HARMFUL INSECTS, UTILIZACAO AND PROCESS FOR the PREPARACAO OF COMPOSICOES 机翻标题: 暂无翻译,请尝试点击翻译按钮。

源语言标题
(BR8600428) Compostos heterociclicos,processo para sua preparacao,composicoes inseticidas,processo para combate a insetos daninhos,utilizacao e processo para a preparacao de composicoes
公开号/公开日
BR8600428 A 1986-10-21 [BR8600428]BRPI8600428 A1 1993-02-16 [BR8600428]BRPI8600428 B1 1998-10-27 [BR8600428] / 1986-10-211993-02-161998-10-27
申请号/申请日
1986BR-0000428 / 1986-02-03
发明人
SHIOKOWA KOZO;TSUBOI SHINICHI;KAGABU SHINZO;MORIYA KOICHI;
申请人
BAYER AGROCHEM;
主分类号
IPC分类号
A01NA01N-033/18A01N-043/00A01N-043/40A01N-043/50A01N-043/54A01N-043/56A01N-043/58A01N-043/60A01N-043/647A01N-043/653A01N-043/66A01N-043/72A01N-043/74A01N-043/76A01N-043/78A01N-043/80A01N-043/82A01N-043/84A01N-043/86A01N-043/88A01N-047/02A01N-047/16A01N-047/22A01N-047/38A01N-051/00A01N-057/32C07DC07D-207/20C07D-207/22C07D-211/70C07D-211/72C07D-213/00C07D-213/61C07D-233/20C07D-233/52C07D-239/06C07D-239/18C07D-263/10C07D-263/28C07D-265/08C07D-277/00C07D-277/10C07D-277/18C07D-279/00C07D-279/06C07D-401/06C07D-401/14C07D-403/06C07D-403/14C07D-405/06C07D-405/14C07D-409/06C07D-409/14C07D-413/06C07D-413/14C07D-417/06C07D-417/14C07D-419/06C07F-009/6558
摘要
(BR8600428) Novel insecticides of the formula in which n is 0 or 1, X is S, O, Y is N or Z is a 5- or 6-membered nitrogen-containing heterocyclic ring, and R to R9 variously represent hydrogen or specified organic radicals.  (From US6022967 A)
机翻摘要
暂无翻译结果,您可以尝试点击头部的翻译按钮。
地址
代理人
代理机构
;
优先权号
1985JP-0018627 1985-02-04 1985JP-0018628 1985-02-04 1985JP-0023683 1985-02-12 1985JP-0106853 1985-05-21 1985JP-0106854 1985-05-21 1985JP-0219082 1985-10-03
主权利要求
(BR8600428)  OF 1155 DEO DEMAND On 1. Heterodolloos composites l oarsotarisados by the fact to present the formula (/) where: n represents or 1, 5. itle 82, 2. 5 represent fte It, independently, a hydrogen atom or a group alquila, 2 3 and 2 4 represents, independently, one &tomo of hydrogen, a group bidroxi or a group alquila, where n represents 1, natio 2 2 can form, a double linking, together with 2 5, X represents a hydrogen atom, one &tomo of oxygen, the following groups: 4-27 or -62-11 8, 2. 7 represent a hydrogen atom, one &tomo of halogenio, a group hidroxi, a group 81-4 a group bensiloxi, a group alquila that it can be substituted by at least a selected substitute if DG dea classroom formed for groups alce* groups alquiltio, a group olmo, atoms of dialquilamino and trialquilsilil halogenio, groups, a group alquenila that it can eer substituted for ua halogenio atom, a group alquinila that it can be substituted by a halogenio atom, a group crack that can be substituted by a group alquila and/or an atom of haloganloom gru po bensila that it can be substituted By me inthe one sUbatituinte dea chosen team classroom forms dea for a group Rutila, a group metoxi, atoms of halogenio, groups halonstila, groups halos.deg.. toxi and a group nitro, a group formal, ua gru po alqueniloarbonila, nm group alquilcarbonila, that it can eer substituted for at least ua I go up tituinte seleoloaado dea classroom formed for groups aloosi, a group fenozi, groups alquiltio and atoms of halogenio, ua group bensoila that po of eer substituted for at least one substituted selected you dea classroom formed for halogenio atoms, groups alquila, groups halometila, groups alcozi, groups baloaloosi and ua group nitro, a group bensiloarbonila that it can be goes up tituido for a group alquila and/or an atom of halogenio, US group alcoxicarbonila that it can be substituted by a halogenio atom, a group alquiltiocarbonila, a group fenorLoarbordla that it can be substituted by at least in substi 55. 55555 DG in and the tuinte dea chosen team classroom formed for ua gru po =tila s a group metoxi, a group halometile, groups halometoxi, atoms of halogenio and one gru po nitro, a feniltiocarboniia group that can be substituted by an atom of halogenio and/or a group alquila, a group bensiloxioarbonila, a group monoalquil- or dialquil-aminocarbonile, a group fenileminocarbonila that it can be subotituido for at least a selected subetituinte dea classroom formed for groups alquile, groups haloalquila and atoms of halogenio, a group bensoilaminocarbonila that it can be substituted, for a group alquila and/or a halogenio atom, a group fenilsulfonilemincoarbonila that it can. to be substituted by a group alquila and/or im er halogenio volume, a feniltio group that can be substituted by a group alquila and/or an atom of halogenio, a group alquilsulfonila that it can be I substituted deo for a halogenio atom, a group fenilsul fonila that it can be substituted by at least a selected subatituinte dea formed classroom, for groups alquila, atoms of halogenio and a group nitro, a group alquilcarbonilmetila, a group fenacila that it can be substituted by an atom of halogenio and/or a group alquila, a group organofosfono, a group orgenotionofos es if CG if Of ell tono, the following groups: -0R 2 - W or. -00-W, W represents a group heterodolloo coa the 5 6 members, contends will pelarmos one heterdatomo stamps ruined dea classroom formed for one &tomo of oxige nio, a Momo of sulfur and an atom of nitroge:. pious, which can be substituted by menCs ua selected substitute dea formed classroom, for &tomos of halogenio, pos groups alquila and gra haloalquila, R and represents one &tomo of hydrogen, um' group alquila, ua group ballot box or a group blessed, - represents a nitrogen atom or I group aeguin you:.6-R 9, R 9 represents a hydrogen atom, a halogenio atom, a group hidroxi, a group alooxl, a group bensiloxi, a group alquila that po4e to be substituted by at least a selected eubstituinte dea classroom formed for &tomos of bae, logenio, a alquiltio group hidroxi, groups alcoxi, pos, me the .deg.lano group, groups mono- or dialquilemino, groups alquilcarbonila, groups alooxioarbonila and groups fenoxioarbonila, umexu po alquenila that it can be substituted by one &.tomo of halogenio, a group alquinila, a group crack that can be substituted by a group ai kilo and/or one &tomo dea halogenio, a group ales quiloarbonila that it can be substituted by a G and Cs 5555. Of 55 halogenio atom, a group alqueniloarbonila. a imburana group that can be substituted by at least a selected aubetituinte dea alasse formed for atonos of halogenio, grouped elquila and groups alooxi, a group alooxioarbonila that it can eer I substituted deo for a halogenio atom, a group elquiltiooarbonila, a group fenoxioarbonila that it can aer substitutes deo for at least a dea selected eubetituinte oily formed for atoms of halogenio, groups alquila, groups alooxi and a group nitro, a group feniltiocarbonila that alquila can be substituted by a group and/or an atom of halogenio, a group feniltiocarbonila that alquila can be substituted by a group and/or an atom of halogenio, a group bensiloxicarbonila, a group beneolleminooarboxila that it can be SUS tituido for a group alquila and/or an atom of halogenio, a group fenileulfonilaminooarbonila that alquila can be substituted by a group and/or an atom of halogenio, a group alquilaulfonilaminooarbonila, a alquiltio group, a group alquileulfonila that it can be I substituted deo for a halogenio atom, a feniltio group that can be substituted by a group alquila and/or an atom of halogenio, In IS : : : : 5: HALF a group fenileulfonila that it can be substituia: deo for a group alquila and/or a mio atom of haloge, alem of this, 8 9 can form a bie-form of fOr mule (1), through a group methylene, R represents a hydrogen atom or a group alquila, and Z represents a group haterodolloo oom the 5 6 members contends at least one heteroatomo in it loved dea classroom formed for a mio atom of oxige, a sulfur atom and an atom of nitrogenid, which can be substituted by "telim a selected substitute dea classroom formed for atoms of halogenio/groups alquila, groups haloalquila, a group nitro, a oiano group, gru pos 820=4 groups alkaline, grouped alquileulfinila, groups alquilsulfonila, grouped alquenila, acilamino group haloalcoxi, groups haloalquiltio, gru poe hnloelquenila, groups, grouped hm, lomoilemlno, groups alooxioarbonila, a group tioolanato, groups alquinila, a group aduo, grouped dialquilemino alquilamino, groups, umgru po oarboxi, a group hidroxi l a group maroapto, groups ololoalquila, a group oxo, a group uncle xo, grouped aloorloarbonilamino haloalqueniltio, groups alcoxialquila, groups, a group 'urbe, mona, groups atila, groups alquileminocarbonila, groups dialquileminocarboalla, a group will be Of. Ga Gil in six 88 if sa in 68 mule, groups anila optionally substituted for substitute selected dea classroom forms dea for atoms of halogenio, groups alquila, gra pos halogenoalquila, groups alcoxi, group ai tro and group damage, groups ariloxl optional mind substituted for substitute as that one presented for groups anila -a l and groups aralquila optionally substituted for the same substitute presented for gru pos armpit, I content that, where R 1, R 2, R 3, 3 4 9 R 5 and R 6 represent, simultaneously, atoms of hidrogenia X represent 4111 and I represents .611, then Z doesnot can indicate the piridil group. 2. Composites, in accordance with claim 1, characterized for the faio of that n represents or the 1, and l and, 5 R and R 6 represent, independently, a hydrogen atom or a group alquila I contend 1 the 4 carbon atoms, R 3 and R 4 you dam has, independently, a hidrogenia atom a group hidrosi or a group alquila I contend 1 the 4 carbon atoms, X represents a sulfur atom, an atom of =Lo b ulo 4, the following groups:.4 2 7 or -12-119 B7 represent a hidrogenia atom a fluor atom, a chlorine atom, a bromine atom, a group bidroxi, a group alcem.  I contend 1 the 4 carbon atoms, a group benziloxi, one gru if GE if if. if DD if Cs if 8. po alquila I contend 1 the 4 carbon atoms that can be substituted by at least one subatitu fight selected dea classroom formed for groups alcoxi contend 1 the 4 carbon atoms, groups alquiltio I contend 1 the 4 carbon atoms, a group olmo, a fluor atom, a chlorine atom, a bromine atom, a dimetilamino group and trimetilsilil, a group alquenila I contend 2 3 atoms of car bono that they can be substituted by a chlorine atom, a group alquinila I contend 2 3 atoms of oar good, a group bensila that it can be substituted by at least a selected substitute dea classroom taken for a group mutilates, az group to toxi l.= fluor atom, a chlorine atom, an atonic one of bromine and a group nitro, a group forni la, a group alquenilcarbonila endowed with one ai quenila I contend 2 3 carbon atoms, a group alquila I contend 1 the 5 atoms daoarbo in what it can be substituted by at least a selected substitute dea classroom become for a group metoxi, ua group fenoxi, an atom of fluor, a chlorine atom and a bromine atom, a group bensoila that it can be substituted by at least a selected substitute dea classroom formed for an atom of fluor, a chlorine atom, a bromine atom, a group mutilates, a group trifluormetila, a group metoxi, a group difluommetozi, a group trifluorometoz1. e a group nitro, a bensilcarbonil group that can be substituted by at least a selected substitute dea classroom formed for a fluor atom, one &te me of chlorine and a bromine atom, a group micoxioarbonila endowed with one alquila I contend 1 the 4 carbon atoms that can be substituted by one &tomo of fluor and/or a chlorine atom a group alquiltiooerbonlla endowed with one elqui la 'I contend 1 the 4 carbon atoms, a group fenozicarbonila that it can be I substituted deo for at least a selected substitute dea classroom formed for a group metila, an atom of fluor, a chlorine atom and an atom of bromine, a group. feniltiocarbonila that it can be substituted by at least a selected substitute dea classroom formed for a group metila, aer fluor volume, a chlorine atom and a bromine atom, a group bensiloxioarbonila, a group dl metilaminooerbonila, a group fenilaminocarboni la that it can be substituted by at least a selected substitute dea classroom formed for a group metila, an atom of fluor, a chlorine atom and a bromine atom, 2. 5 a group bensolleminocarbonila that it can be I go up tituido for at least a substitute eeleolon ado dea classroom formed for a group =til% an atom of fluor, one &tomo of chlorine and one &tomo of bromine, a group fenileulfonilaminocarbonila that it can be substituted by at least a subetituinte, dea chosen team classroom formed for one &tomo of fluor, a chlorine atom and a bromine atom a feniltio group, a group alquileulibmila that it can be substituted by one &tomo of fluor and/or one &tomo of chlorine, a group fenileulfonila that it can be substitutes 'deo for at least a selected substitute of classroom formed for a group metila, one &tomo - of fluor, one &tomo of olor: N.um &tomo of bromine, and a group nitro, ua group metiloarbonilmetile, a group fenaoila that it can be substituted by an atom to rhyme and/or one &tomo of chlorine, a group 'organofoefono, a group organotionofosfono, the following groups: -02 2 - W or -00-W, W represents a group heterodoliao contends the 5 6 members one or two endowed with betero&tomos chosen teams dea classroom formed for a &tono of oxygen, one &tomo of sulfur and a trogenio atom of ni, which can be substituted by at least a selected eubstituinte dea classroom will be n ada for one &tomo of fluor, one &tomo of chlorine in 55 5 in. e 5. and to a and and 5 to the o to eme 11. in it joins the n il and me .deg. and n e: 5:59 5 85 5 me the atom of bromine and groups alquila I contend 1 the 4 carbon atoms, 2., it represents in the hydrogen atom, a group alquila I contend 1 the 4 atoms of. oarbone, a Zunia group or a group bensila, Y represents a nitrogen atom or it I group it followed you:.0-11 9, R, represent a hydrogen atom, a fluor atom, a chlorine atom, ua bromine atom, a group hidroxi, a group alooxi contend 1 the 4 carbon atoms, in the group bensiloxi i - one gru po alquila I contend 1 the 4 carbon atoms that can be substituted by at least one eubstitu inte selected olaese Sornada for an atom of troar dea, a chlorine atom, a group hidrosi a group aloosi I contend 1 the 2 carbon atoms, groups alquiltio I contend 1 the 2 carbon atoms, ua group swan, a dimetilemino group, grupod alquiloarbonila I contend 1 alquila with 1 the 2 carbon atoms and groups alcoxioaflonila, I contend one alquila with 1 the 2 carbon atoms, 2. 5 a group alquenila I contend 2 3 atoms of oar boron, a group crack, a group alquilcarbonila I contend one alquila coa 1 the 4 carbon atoms that can be Inlaid tuteio for at least a substitute select . 12 deo deo group become for a group =taxi, an act to the one of chlorine, and a fluor atom, a group alqueniloarbanila I contend one alqueni la coa the 2 3 carbon atoms, a group bensofla that it can be substituted by at least a eeleolonado substitute dea classroom formed for a fluor atom, a chlorine atom, went bromine atom, a group metozi and a group instila, a group alcorioarbonila that it can be substitutes deo for a fluor atom and/or an atom of olorq a group alquiltiocarbonila I contend one alquila with 1 the 4 carbon atoms, a group fenozioarbonila that it can be substitutes deo for it flowed a selected subatituinte dea olaeee formed by a fluor atom, an act to the one of chlorine, a bromine atom, a group mutilates, a group =tont and a group nitro, 1. 5 a group feniltiocarbonila, a group bensiloxi, carbonila, a group bensolleminocarbonila that ensebe tituido by at least one can substitutute selected dea classroom formed for a group =tilas an atom of fluor, a chlorine atom and a bromine atom, 2. 5 a group alquileulfonilaminocarbonila contends one alquila with 1 the 4 carbon atoms, a alquiltio group Dipping in grease 1 the 4 atoms of oar 550. 56 IS 55 511 i 55 55 IS 8. 1 8 9 I: 0: : 5 I 5 G I 5 5 5 I 5 M5O 5 II 5 CP 5 C C 55 IS 5 5 11 5 Me 59 ITSELF 55 5 550 55 - 1 3 bono, a group alquileulfonila that it can be substitutes deo for ua &tomo of fluor and/or one &tomo of clearly, a feniltio group that can substitute for 5. at least a selected subetituinte dea alasse formed for a group mutilate, a dafluor atom, a chlorine atom and one &tomo of bromine, or a group fenileulfonila that it can be substituido by at least a selected eubetituinte dea classroom formed for a group metila, one &tomo of fluor, a chlorine atom and one &tomo of bromine, moreover $ 9 can form one bis-lines of formula (i), through a group methylene, represents a hydrogen atom or a group you mutilate and IS represents a group beteroololiod contends the 5 6 hatero&tomos members endowed with one trile ee lecionados dea classroom formed for one &tomo of oxygen, one &tomo of sulfur and a troganio atom of ni, which can be substituted by at least a selected subatituinte dea classroom will be swims for a fluor atom, one &tomo of chlorine one &tomo of bromine, groups alquila I contend 1 the 4 carbon atoms that can be substituted by one &tomo of fluor and/or a chlorine atom, a group nitro, a group top of a mountain, groups alquilsulfinila I contend 1 the 4 &tomos of carbon, Gives IS 5. ME O IS -14grupos alquileulfonila I contend 1 the 4 carbon atoms, groups alcosi I contend 1 the 4 carbon atoms, that can be substituted by an atom of flu- 5: and/or a chlorine atom, groups alquiltio I contend 1 the 4 atoms of Garbo in what an atom of fluor and/or a chlorine atom can be substituted by, groups alquenila I contend 2 3 atoms of Garbo in what they can be substituted by a chlorine atom, a group -temida that can be substituted by a fluor atom e/on a chlorine atom, groups alooxicarbonila I contend one alquila with 1. 5 1 the 4 carbon atoms, a group tiocianato, grupoe alquinila I contend 2 4 atoms of Garbo in, a group amimo, a metilamino group, a dimetilamino group l. a group -atila, a group fornila, a group oarboxi, a group bidroxi l ua group meroapto, groups ololoalquila I contend 3 7 carbon atoms, one grgpo oxo, alqueniltio a Lame group, groups substituted by a fluor atom, a chlorine atom and/or a bromine atom, groups alooxialquila I contend 2 4 carbon atoms in the total, groups elquileminooarbonila I contend one alquila oom 1 the 2 carbon atoms, in Del In Itself 0 5 0 Ill G GE It is *G and II IP MI - the 35 0 groups dielquileminocarbonila I contend one alquila with 1 the 2 carbon atoms, a group it repels, a group fenoxi and a group ben day, I content that where 2 1 1 12 2, 11 3, 2 4, 8 5 and 86 5 represent, simultaneously, atomoe'de hidroge aio, represents - NH, and Y representa.02 1 then 8 does not have to indicate the piridil group. 3. Composites, in agreement coa claim 1, characterized for the fact of that n represents or 1, 1. 9 2 9 8 5 and 8! * they represent, indeuendentemente, a hydrogen atom or a group metila, 8. 3 and 2 4 represents, independently, an atom of hidrogenio or a group metila, represents a sulfur atom, an atom of 'exempt or the following groups: 4-2 7 or -0511-2P 2 7 represent a hydrogen atom, a group alquila that it can be substituted by at least a selected subetituinte dea formed classroom, for a group matoxi, a group etoxi, a group Jingled a etiltio group, a group (damage, a fluor atom, a chlorine atom, and a group trimetile1111, a group alila that it can be substituted by a chlorine atom, a propargil group, a group bensila that it can be would substitute for the 16. a group mutilates and/or one &tomo of chlorine, a group tonna, a group viniloarbonila, ua group alquilcarbonila I contend one alquila, with 1 the 3 &tomos of carbon that it can eer I inlaid tuido for at least a eubstituinte select dea deo classroom formed for ua group alatoai, a group fenoxi and a chlorine atom, a group benzoila that it can eer substituted per at least a selected substitute dea days, if formed for one &tomo dea chlorine, ua bromine atom, a group mutilates, a group trifluorometl la, ua group metoxi and a group nitro, ua group bensilcarbonila that it can eer substitutes deo for a chlorine atom, 1. 5 a group alooxioarbonila contends one alquila, with l'a 2 carbon atoms that can be eubeti coupon stub for one &tomo of fluor elou one chlorine atom, a group alquiltiooarbonila I contend joins alquila oom 1 the 2 carbon atoms, a group fenoxioarbonioa that it can be substitutes deo for a Rutila group and/or a chlorine atom, a group feniltiooarbonila that it can be substituido by one &tomo of chlorine, a group bensiloxicarbonila, a group to dimettlar minooarbonila, a group fenileminocarbonila, a group benzolleminocarbonila, a group fenileulfonileminocarboni1a that it can Of le if DG GE - 1 7 to be substituted by a put group and/or one &te me of chlorine, a feniltio group, a group metileulfanila that it can be substituted by one &tomo of chlorine, a group fenileulfonila that it can be substituted by a group mutilates, a group metilosztonilmetila, a group fenaoila that it can be substituted by a chlorine atom, a group 0,0-dietiltionofoefono, a group 0-et11-13-n-propiltiolofoefono, the following groups: -011 2 -7 or -00-7, W represents a group heterodolloo with 5 the 6 members contends one or doia we heteroltemos stamps olonados dea classroom formed for one &tomo of oxygen, one &tomo of sulfur and one &tomo of nitrogen, which can be substituted by one &tomo of in one, one &tomo of chlorine, a bromine atom, 1. 5 and a group mutilates, R represents it one &tomo of hydrogen, a group put, a group: anila or a group banana, Y represents one &tomo of nitrogen or I group seguin you:.0-p 9 r and R 9 represents one &tomo of hydrogen, a chlorine atom, one &tomo of bromine, a group hidroxi a group metoxi, a group bensiloxi, a group alquila that it can be substituted by at least if Cs - 18 a seleoionado substitute dea classroom baking for a fluor atom, a chlorine atom, a group hidroxi, a group metoii, a group ciam, a dimetilemino group, a group acutila and a group metoxioarbonila, a group alila, a group fenila, a group agglutinates that it can be substituted by a chlorine atom, a group viniloax, bonila, a group alilcarbonila, a group benzoLla, a group alcoricerbonila I contend one alquila coa 1 the 2 atoms de'oarbono that it can be I struck tuido for a fluor atom, a group n-butiltiooarbonila, a group fenoxi oarbonila that it can be substituted by a chlorine atom s and/or a group mutilates, a group funnel tiocarbonila, um'grupo benziloxicarbonila, a group beasoileminocarbonila that it can be arabuta, tuido for an atom of chlorine, a group fenilsulfonileminocarbonila that it can be substituted by a group mutilates, 1. 5 in the group metileulfonileminocarbonila, a propiltio group, a group metileulfonila that it can be substituted by an atom of fluor and/or a chlorine atom, a feniltio group that can be substituted by a chlorine atom, or a group fenileulfonila, moreover, R 9 can form bis - form of fOr mule (i), through in the group mutilates, COMPACT DISC 55 DG GD IN and 19. Of cm ITSELF 5555 DEO represent one &tomo of hydrogen or one groups mobila i and Z represents a bateroololico group contends the 5 6 members endowed with one it harnesses bateroatomos if 5. lecionados dea classroom formed for one &tomo of osinalo, a sulfur atom and one &tomo of nitrogenio, being that at least one of them it is a air nitrogenio volume, which can be substituted by the monos 10 a selected substitute dea. classroom formed for an atom of Mor, an atom of chlorine, one homodebromo, a Estila group, groups fluoroalquila I contend 1 the 2 carbon atoms, a group metoxi l a metiltio group, a group me 15. tilsulfinila, a group metileulfonila, a group nitro, a group top of a mountain, a group trifluorometoxi, a trifluorometiltio group s, a group alila, a -temida group, a group metoxicarbonila, a group aoetila, a group formila and a group 20 pair. boxila l contanto that, where al, 3 2, R 3, E1 4, 3 5 and 6 R re prefeel, simultaneously, &tomos of bidroge mio, I (represent -61 and Y representa.121 1 then: 5 25 do not have to indicate the piridil group. 4. Compound 3- (2-chlorine-5-pirldilmet11) - 2 (nitro matileno) tetrehidro-25-1,3-tiasina, in accordance with the king vindications 1 the 3, characterized for the fact of being repre. HOLLOW DG CG 5 OF SC 8. G MC G CGD. GC. GE G GO. MD WIN seated for the following formula: (:)e, OHNO 2 0. E 2 - -01 5. Compound 3- (2-oloro-3-piridilmetil) - 2- (nitro methylene) tiazolidina 9 in agreement, with claims 1 the 3, characterized for the fact of being represented by if the 5 gaiata formula: E>011/10 2 Ilir - CL 6. Compound 3- (2-fluoro-5-pirldilmet11) - 2- (ai trometileno) tetrahidro-22-1,3-tiazina one, in accordance with claims 1 the 3, characterized for the embryo dg to be represented by the following one nullified: 7. Compound 3- (2-fluoro-3-piridilnetil) - 2- (nitroaetileno) tiazolidina 9 in accordance with claims 1 the 3, characterized for the fact of being represented by the following formula: I read to 5 1 co G and 21. 8. Compound 3- (2-bromine-5-piridilmetil) - 2- (ni trometileno) tetrehidro-28-1 1 3-tiazina, in agreement coe claims 1 3 1 oaraoterizado by the fact of being represented by the following formula: C R NOHNO 2 011. 5. 9. Compound 3- (2-bromine-3-piridilmetil) - 2- (nitro methylene) tiazolidina one, in accordance with ae reivindica95es 1 the 3, characterized for the fact of being represented by if you guided CH 2 - 10. Compound 3-C1- (2-chlorine-5piridil) etil7=2 10 (nitromatileno) tiazolidina l in accordance with demands them coes 1 the 3, characterized for the fact of being represented by the following formula: i 9 I I d - 22. 4. read ITSELF. E>000 2 3. C-Gil- - ai 11. Compound 3- (2-gmetal-5-pirldilmetil) - 2- (ni trometileno) tiesolidina one, in accordance with claims 1 the 3, characterized for the fact of being represented by the following formula: 11. : >CHNO 2 CEr 12. Compound 3- (2-metal-5-piridilmetil) -2- (ni trometileno) tetrehidro-28-1,3-tiazina l in accordance with claims 1 the 3, characterized for the fact ds to be represented by the following formula: 13. Compound 3- (2-trifluoromet11-5-piridilme til) - 2- (nitrometileno) tiazolidina one, in accordance with claims 1 the 3, characterized for the fact of being representadopela following formula: DG DD - me and 5155 23e z eme ee ee ee Lh02 2 Lh 0 0E 2 - 14. Compound the 3- (2-etil-3-pirldilmetil) - 2- (nitro methylene) tiasolidina, in accordance with ae claims 1 the 3, caracterizadn'por the fact of being represented by if guinte formula: -0 2 and 5. 15. Compound 3- (3-pirldilmet11) - 2- (nitrometileno) tetrahldro-28-1,3-tiasina one, in accordance with claims 1 the 3, characterized for the fact of being represented by the following formula: 16. Compound 1- (5-pirasolilitetil) - 2- (nitrozaciti, leno) laidasolidina one, in accordance with claims 1 the 3., characterized for the fact of being represented by the following formula: - "ne n if 17. Compound 1- (3-oloro-1-net11-3-pirazolilme t11) - 2- (altrometileno) imidazolidiaa, in accordance with ae claims 1 the 3, characterized for the fact of being represented by the following formula: 18. Compound 1- (1-I put],--pirazolilmetil) - 2.4ni trometileno) tetrahidropirimidina, in accordance with ae claims 1 the 3, characterized for the fact of being represented by the following formula: 19. Compound 1- (1-metal-4-pirazolilmetil) - 2- (ni IS MG MD . 25 one ee tronetileno) igidazolidina, demands in accordance with them. ;  Oes 1 the 3, characterized for the fact of being represented by the following formula: 20. Cogposto 1 - (3-triflncronetil-5-isoznsolilne 5. til) - 2- (nitrOmatileno) tetrahidropirimidina one, in agreement;  with claims 1 the 3, characterized for the fact of being represented by the following formula: 21. Conpoeto 1- (3-metal-3-isoxazolilzietil) -2 - (nitrometileno) inidazolidina one, in agreement coa reivindi- 10 .deg.acoes 1 the 3, characterized for the fact of being represented by following fOraula: ... s DG to the O - 26 - 5 you 1115 and" 0 2 CH2- 22. Compound 1.43-met11-3-leorazolilizet11) -2 - (nitrometileno) tetrahldropirimidina 9 in accordance with es claims 1 the 3, characterized for the fact of being represented by the following formula: 23. Compound 1- (5-leo-ozszolilmet11) - 2- (altrome tileno) imidazolidina l in accordance with claims 1 the 3, the characterized for the fact of being represented by if guinte formula: 24. Compound 1- (2.met11-5-tiaiolilmetil).2. (21. trometileno) imidazolidina, in accordance with it demands them - G ile I n 5 ne j and 5 5 8 u and g and I I and S I AND I I D g If 5 1 1 1 1 45 and 95 55 goes 1 the 3, characterized for the fact of being represented by the following formula: 25. Coapoeto 1- (2-oloro.5.tiazolilmatil) - 2- (nitrometileno) tetrehidropirialdina one, in accordance with ae king vindicagace 1 the 3, characterized for the respected fact of ser'reprea for the following formula: 01. 26. G: tax 1- (2-trifluoromet11-5-tiazolilmetil).2. (nitrometileno) imidazolidina, in accordance with claims 1 the 3, characterized for the fact of being re, preeentado for the following formula: e 5 8 11: : : :.: - au Of 27. Compound 1- (1 9 2 9 5-tiadiazol-30.11metil) -2 - (nitrometileno) tetrehidropirimidina l demands in accordance with them: 35es 1 the 3, characterized for the fact of being represented by the following formula: T1 5,423110 2 ollr ic 28. Compound 1- (1 9 2 9 3-tiadiazol-3-11metil) -2 - (nitrometileno) tetrabldropirizidina l in accordance with reivindicagaes 1 the 3, characterized for the fact of being represented by the following formula: 29. Compound 1- (2-metil-5-tiasolilmetil) - 2- (nitrametileno) tetrablaropirimidina one, in agreement coa the king vindications 1 the 3, characterized for the embryo of being represented by the following formula: CHNO 2 C1 2 - ,1 IS CO Ia : Z: : : 29 0 112 5 ei n and ei n and I n 605 55 1: 18 30. Compound 1- (2-oloro-5;  41azolilmetil) - 2- (ni= trometileno) imidazolidina one, in accordance with demands them gane 1 the 3, characterized for the fact of being represented by the following formula: 01. 5. 31. Compound 1. (5-tiazolilmetil) - 2- (nitrometlle in) tetrahidtopirimidina one, in accordance with claims 1 the 3, characterized for the fact of eer represented for the following formula: 32. Compound 1- (5-piriaidinilmet11) - 2- (nitrome- 10. tileno) imidazolidina l in accordance with claims 1 the 3, characterized for the embryo of being represented by the following formula: Itself - 30.y 33. Compound 1- (2-metal-5-pirinidinilnetil) -2 - (nitrometileno) inidasolidina one, in accordance with es reivindicaoSee 1 the 3, characterized for the fact of being represented by the following formula: 5. 34. Compound (- (2-pirazinilmetil) - 2- (nitrometilano) inidazolidina one, in agreement coa ae reivindicacaes 1 the 3, characterized for the fact of being represented by the following formula: 35. Compound 1- (3-metal-2-pirazinilmet11) - 2- (ai 10 trometileno) imidazolidina one, in accordance with demands them gaes 1 the 3, characterized for the fact of being represented by the following formula: itself Of GE if and and n and I n e: : G and n and theses if 36., Compound 1. (2-cloro.5.pirimidinilmetil) -2 - (nitrometileno) tetrahidropirimidina one, in agreement coa reivindicagBee 1 the 3, characterized for the fact of being represented by the following formula: C H), 011/10 2 011. 2 -0-01 37. Compound 1- (2-cloro.5-pirimidinilnetil) -2 - (nitrametileno) imidazolidina g in agreement oan reivindi- .deg.agaloe 1 the 3, characterized for the fact of being represented by the following formula: - 5 TOP OF A MOUNTAIN 2 01. 2 - C5 - CH 3 38. Compound 1- (2--chlorine-3-piridilmetil)--2- (21 trometileno) tetrahidropirimidina, in accordance with the king vindications 1 the 3, characterized for the fact of (...)
法律状态
(BR8600428) LEGAL DETAILS FOR BR8600428  Actual or expected expiration date=2006-02-03    Legal state=DEAD    Status=REVOKED     Event publication date=1986-02-03  Event code=BR/APP  Event indicator=Pos  Event type=Examination events  Application details  Application country=BR BR8600428  Application date=1986-02-03  Standardized application number=1986BR-0000428     Event publication date=1986-10-21  Event code=BR/A  Event type=Examination events  Published application  Publication country=BR  Publication number=BR8600428  Publication stage Code=A  Publication date=1986-10-21  Standardized publication number=BR8600428     Event publication date=1993-02-16  Event code=BR/A1  Event indicator=Pos  Event type=Examination events  Published application  Publication country=BR  Publication number=BRPI8600428  Publication stage Code=A1  Publication date=1993-02-16  Standardized publication number=BR8600428     Event publication date=1995-12-12  Event code=BR/FB19  Event indicator=Neg  Event type=Event indicating Not In Force  Grant procedure suspended (art. 19) Suspensao do andamento do pedido (art. 19)    Event publication date=1998-02-25  Event code=BR/FF  Event indicator=Pos  Event type=Event indicating In Force  Decision: granting Decisao: deferimento    Event publication date=1998-10-27  Event code=BR/B1  Event indicator=Pos  Event type=Event indicating In Force  Granted patent / Granted pipeline patent  Publication country=BR  Publication number=BRPI8600428  Publication stage Code=B1  Publication date=1998-10-27  Standardized publication number=BR8600428     Event publication date=1998-10-27  Event code=BR/FG  Event indicator=Pos  Event type=Event indicating In Force  Letter patent granted Carta de patent expedida    Event publication date=2004-08-10  Event code=BR/B25D  Event type=Change of name or address  Event type=Reassignment  Requested change of name of applicant approved Notificacao do deferimento da alteracao de nome requerida    Event publication date=2012-12-04  Event code=BR/B21A  Event indicator=Neg  Event type=Event indicating Not In Force  Expiry acc. art. 78, item i of ipl- expiry of the term of protection Extincao de patente e certificado de adicao de invencao: extincao - art. 78 inciso i da lpi PATENTE EXTINTA EM 27/10/2008
专利类型码
AA1B1
国别省市代码
若您需要申请原文,请登录。

最新评论

暂无评论。

登录后可以发表评论

意见反馈
返回顶部