Benzoylderivate, procedures for their production and their use as herbicides and plant growth modulators 机翻标题: 暂无翻译,请尝试点击翻译按钮。

公开号/公开日
DE19840337 A1 2000-03-09 [DE19840337] / 2000-03-09
申请号/申请日
1998DE-1040337 / 1998-09-04
发明人
ALMSICK ANDREAS VAN;WILLMS LOTHAR;AULER THOMAS;BIERINGER HERMANN;ROSINGER CHRISTOPHER;
申请人
HOECHST SCHERING AGREVO;
主分类号
IPC分类号
A01N-043/18A01N-043/40A01N-043/50A01N-043/54A01N-043/56A01N-043/60A01N-043/80A01N-057/12A01P-013/00C07D-333/56C07D-335/06C07D-335/16C07D-409/04C07D-409/06C07D-409/12C07D-409/14C07D-413/12C07D-413/14C07D-417/12C07D-417/14C07F-009/09C07
摘要
(DE19840337) The invention relates to benzoyl derivatives of general formula (I), to a method for producing them and to their use as herbicides and plant growth regulators.  In said general formula (I), R<1>, R<2>, R<3>, R<4> and R<5> represent different organic radicals, Q represents an isothiazole, isoxazole, cyclohexanedione or beta -ketonitrile radical and A, B, E and X represent mono- or polyatomic divalent units.
机翻摘要
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地址
代理人
代理机构
;
优先权号
1998DE-1040337 1998-09-04
主权利要求
(DE19840337) 1. Benzoyl derivatives of the formula (I),  wherein Q is a radical of the formula (II), (III) or (IV)  R1, R2, R3 independently hydrogen, Hydroxy, Thio, amino, cyano, nitro, Halogen or an optionally substituted hydrocarbon radical, which may contain one or more, identical or different heteroatoms such as oxygen, sulfur, nitrogen, fluorine, chlorine, bromine and iodine includes; R4 hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, Phenyl, optionally substituted by one or more said six lastmentioned groups, identical or different substituents selected from the group consisting of Halogen, nitro, cyano, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy and alkylthio substituted; R5 optionally mono - or polysubstituted by identical or different substituents substituted Heteroaryl, cycloalkyl or aryl; A A divalent moiety selected from the group O, S, so, so2, noa, chra and cra Rb ; B A saturated or one or more multiple bonds and one to four carbon atoms existing chain containing, optionally substituted with alkyl, halo, alkoxy, haloalkoxy or an optionally substituted with alkyl, halo, alkoxy, haloalkoxy, Halogen, cyano or nitro-substituted Phenyl radical is substituted; E is A bond, A saturated or one or more multiple bonds formed of one to six-containing divalent group C units, crc, crc Rd, N, nrc, S, so, so2, O and co; O X from A divalent moiety, S and nre ; R6 alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, cyano, cyanato, thiocyanato, Halogen or orf ; A divalent moiety selected from the group O Y, S, nh, N-alkyl or chr7 ; R7 hydrogen, Tetrahydropyran 3-yl, Tetrahydropyran 4-yl, Tetrahydrothiopyran 3-yl, alkyl, cycloalkyl, alkoxy, alkoxyalkyl, alkylcarbonyl, alkoxycarbonyl, alkylthio, Phenyl, wherein the hydrocarbon portion of the eight last-mentioned radicals substituted with one or more, identical or different substituents selected from the group consisting of Halogen, alkoxy and alkylthio substituted, or  two R groups attached to a common atom7 form a chain of the group OCH2 CH2 O, OCH2 CH2 CH2 O, sch2 CH2 S and sch2 CH2 CH2 S, which is optionally substituted by one to four methyl groups, or two R groups on adjacent carbon atoms directly bonded7 carrying them form a bond or an optionally substituted 3 together with the carbon atoms to 6-membered ring; Z is a bond, a divalent moiety selected from the group O, S, so, so2, NH, N-Alkyl or chr7, wherein Y Z is intended to mean a divalent moiety and at the same time, as an oxygen link, nitrogen or sulfur atom; G1 -G2 a divalent moiety selected from the group ocr9, scr9 and no10 Cor11, wherein the linkage is to be performed with the ring system is, that the carbon atom through each of these divalent ring system a percentage of a double bond; R8 hydrogen, Alkyl or Alkoxy-carbonyl; R9 hydrogen, Alkyl, Cycloalkyl, haloalkyl or halocycloalkyl; R10 hydrogen, Alkyl, Alkenyl, alkynyl, Cycloalkyl, Phenyl, Benzyl, substituted by one or more said six lastmentioned groups, identical or different substituents selected from the group consisting of Halogen, Cyano, nitro and Alkoxy substituted; R11 hydrogen, Formyl, Alkyl, halo, or group L-R alkoxvalkxl12 ; a divalent moiety selected from the group so L2, Co, chrg Co or Crg Rh ; R12 Alkyl, halogenoalkyl, Alkoxy, haloalkoxy, Alkyl amino, Dialkylamino, Cycloalkyl or substituted with one or more, the same or different radicals from the group consisting of Cyano, nitro, Alkyl, Alkoxy, halkoalkyl and haloalkoxy-substituted Phenyl; Ra and Rb independently hydrogen, Halogen, Cyano, nitro, Formyl, Alkyl, Cycloalkyl, Alkenyl, alkynyl, Alkyl carbonyl and alkylsulfonyl, wherein the hydrocarbon radicals substituted with one or more of the six lastmentioned, identical or different substituents selected from the group consisting of Halogen, nitro, Cyano, Alkyl, Cycloalkyl, Alkenyl, alkynyl, Alkoxy and alkylthio substituted; Rc and Rd independently hydrogen, Halogen, nitro, Cyano, Alkyl, halo, Cycloalkyl, Alkenyl, haloalkenyl, alkynyl, haloalkenyl, Alkoxy, haloalkoxy, alkylthio, haloalkylthio, carbonyl, haloalkylcarbonyl, Alkoxycarbonyl, halo Alkoxycarbonyl, amino carbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkylcarbonyl, carbonyl, haloalkylcarbonyl amino, carbonyl-N-Alkyl amino, alkylsulfonyl, alkylsulfinyl, alkylsulfonylamino, haloalkylsulfonyl, haloalkylsulfinyl, alkylsulfonyl N-alkylamino aryloxycarbonylsmino and; Re hydrogen, Formyl, Alkyl, Cycloalkyl, Alkenyl, alkynyl, Alkyl carbonyl and alkylsulfonyl, wherein the hydrocarbon portion of the six lastmentioned groups optionally with one or more, identical or different substituents selected from the group consisting of Halogen, nitro, Cyano, Alkyl, Cycloalkyl, Alkenyl, alkynyl, Alkoxy and alkylthio may be substituted; Rf hydrogen, Alkyl, halo, Alkoxy, Formyl, carbonyl, Alkoxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkylsulfonyl, haloalkylsulfonyl, Benzoyl or Phenylsufonyl, wherein the concentration of the latter two groups are optionally substituted by one or more, the same or different radicals from the group consisting of Alkyl, halo, Alkoxy, haloalkoxy, Halogen, Cyano and nitro substituted; Rg and Rh independently hydrogen or Alkyl; N 0, 1, 2 or 3; 1 or 2 v; w 0, 1, 2, 3 or 4 are, with the proviso, in R5 Aryl is not Phenyl, when G1 in G1 -G2 E is methylene and sulfur. 2. Benzoyl derivatives according to claim 1, wherein R1, R2, R3 independently hydrogen, Alkyl, Alkenyl, alkynyl, Cycloalkyl, Cycloalkenyl, cycloalkylalkyl, Cycloalkyl Alkenyl, cycloalkylalkynyl, Aryl, Aryl Alkyl, arylalkenyl, arylalkynyl, Heteroaryl, heteroarylalkyl, heteroarylalkenyl, heteroarylalkynyl, Heterocyclyl, heterocyclylalkyl, heterocyclylalkylenyl, heterocyclylalkynyl, Hydroxy, Alkoxy, alkenyloxy, alkynyloxy, Cycloalkoxy, cycloalkylalkoxy, cvcloalkvl alkenyloxy, alkynyloxy cvcloalkvl, cycloalkenyloxy, aryloxy, arylalkoxy, Aryl sulfonyloxy, Aryl alkynyloxy, heteroaryloxy, heteroarylalkoxy, Heteroaryl alkenyloxy, alkynyloxy Heteroaryl, heterocyclyloxy, heterocyclylalkoxy, Heterocyclyl alkenyloxy, alkynyl Heterocyclyl-oxy, Thio, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, alkylthio ;b, alkenylthio ;b, cycloalkylalkynyl Thio, cyclo alkenylthio, arylthio, arylalkylthio, arylalkenyl Thio, Aryl alkynylthio, heteroarylthio, Heteroaryl alkylthio, alkenylthio Heteroaryl, heteroarytatkynyt Thio, heterocyclic Thio, heterocyclic alkylthio, alkenylthio Heterocyclyl, Heterocyclyl alkynylthio, Amino, optionally substituted Mono - or Dialkylamino, optionally substituted Mono - or Diarylamino, optionally substituted Mono - or Di-heteroarylamino, optionally substituted N-Alkyl-N-arylamino, optionally substituted N-Alkyl-N-heteroarylamino, alkenylamino, alkynylamino, cycloalylamin, cycloalkenylamino, Heterocyclyl alkylamino, heterocyclylalkylenyl Amino, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, cycloalkylalkylsulfonyl, alkenylsulphonyl ;b, cycloalkylalkynyl sulfonyl, Aryl sulfonyl, Aryl sulfonyl, Aryl alkenylsulphonyl, arylalkynyl sulfonyl, heteroarylsulfonyl, Heteroaryl Alkyl sulfonyl, Heteroaryl alkenylsulphonyl, heteroarytatkynyt sulfonyl, heterocyclylsulphonyl, heterocyclylaminocarbonyl, alkenylsulphonyl Heterocyclyl, heterocyclylalkynyl sulfonyl, sulfinyl, alkenylsulfinyl, alkynylsulfinyl, Cycloalkyl sulfinyl, ;b alkylsulfinyl, alkenylsulfinyl cvcloalkvl, alkynylsulfinyl cvcloalkvl, arylsulfinyl, Aryl Alkyl sulfinyl, Aryl alkenylsulfinyl, alkynylsulfinyl Aryl, hetero arylsulfinyl, alkylsulfinyl Heteroaryl, heteroarylalkenyl sulfinyl, phenylsulfinyl heteroarytatkynyt, Heterocyclyl sulfinyl, Aryl Alkyl sulfinyl, phenylsulfinyl heterocyclylalkylenyl, Heterocyclyl alkynylsulfinyl, aminosulfonyl, optionally substituted Mono - or dialkylaminosulfonyl, aminosulfonyl optionally substituted Mono - or Di, optionally substituted Mono - or Di-heteroarylaminosulfonyl are, optionally substituted N-Alkyl-N- arylaminosulfonyl, optionally substituted N-Alkyl-N-heteroarylaminosulfonyl are, alkylsulfonyloxy, phenylsulfonyloxy Alkenyl, alkynyl sulfonyloxy, cyclo Alkyl sulfonyloxy, alkylsulfonyloxy ;b, sulfonyloxy ;b Alkenyl, alkynyl sulfonyloxy cvcloalkvl, arylsulfonyloxy, alkylsulfonyloxy Aryl, aralkyl sulfonyloxy, arylalkynyl sulfonyloxy, Heteroaryl sulfonyloxy, alkylsulfonyloxy Heteroaryl, heteroarylalkenyl sulfonyloxy, phenylsulfonyloxy heteroarytatkynyt, sulfonyloxy Heterocyclyl, heterocyclylalkyl sulfonyloxy, phenylsulfonyloxy heterocyclylalkylenyl, heterocyclylalkynyl sulfonyloxy, aryloxycarbonylsmino, alkenylsulphonyl Amino, sulfonylamino alkynyl, Cycloalkyl sulfonyl Amino, Cycloalkyl Alkyl sulfonic Amino, Amino Alkyl alkenylsulphonyl, cycloalkylalkynyl sulfonylamino, arylsulfonylamino, isopropylsulfonylamino Aryl, arylalkenyl sulfono-Amino, sulfonylamino arylalkynyl, heteroarylsulfonyl Amino, Heteroaryl isopropylsulfonylamino, heteroarylalkenyl sulfono-Amino, sulfonylamino heteroarytatkynyt, alkylsulfonyl N-alkylamino, alkenylsulphonyl-N-alkylamino, alkynylsulfonyl-N-alkylamino, cycloalkylsulfonyl-N-alkylamino, cylcoalkylalkylsulfonyl-N-alkylamino, Cycloalkylalkenylsulfonyl-N-alkylamino, Cycloalkylalkinylsulfonyl-N-alkylamino, arylsulfonyl N-alkylamino, heteroarylsulfonyl-N-alkylamino, Arylalkylsulfonyl-N-alkylamino, Heteroarylalkylsulfonyl-N-alkylamino, arylalkenyl sulfono Amino, heteroarylalkenyl sulfono Amino, Arylalkinylsulfonyl-N-alkylamino, Heteroarylalkinylsulfonyl-N-alkylamino, heterocyclylsulfonyl-N-Alkyl Amino, sulfo-heterocyclylalkyl, Heterocyclylalkenylsulfonyl-N-alkylamino, Heterocyclylalkinylsulfonyl-N-alkylamino, carbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, Cycloalkyl-Alkyl, acyl ;b, cycloalkylalkynyl carbonyl, Aryl carbonyl, Aryl Alkyl carbonyl, alkenylcarbonyl Aryl, arylalkynyl carbonyl, heteroarylcarbonyl, heteroarylalkylcarbonyl, heteroarylalkenyl, heteroarytatkynyt carbonyl, heterocyclylcarbonyl, heterocyclylalkylcarbonyl, heterocyclylalkylenyl, heterocyclylalkynyl carbonyl, Carboxyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkoxycarbonyl, cycloalkylalkoxycarbonyl, Cycloalkyl-lower alkenyloxy, alkynyloxy Cycloalkyl carbonyl, aryloxycarbonyl, arylalkoxycarbonyl, Aryl carbonyl alkenyloxy, alkynyloxy carbonyl Aryl, heteroaryloxycarbonyl, heteroarylalkoxycarbonyl, Heteroaryl-lower alkenyloxy, alkynyloxy carbonyl Heteroaryl, heterocyclyloxycarbonyl, heterocyclylalkoxycarbonyl, alkenyloxycarbonyl Heterocyclyl, Heterocyclyl alkynyloxy carbonyl, Amino carbonyl, optionally substituted Mono - or dialkylaminocarbonyl, optionally substituted Mono - or diarylaminocarbonyl, optionally substituted Mono - or Di- Heteroarylaminocarbonyl, optionally substituted N-Alkyl-N- arylaminocarbonyl, optionally substituted N-Alkyl-N- Heteroarylaminocarbonyl, optionally substituted alkylcarbonylamino, substituted or unsubstituted alkylcarbonyl-N-Alkyl Amino, substituted or unsubstituted arylcarbonylamino, substituted or unsubstituted Aryl carbonyl N-arylamino, Amino optionally substituted Heteroaryl, optionally substituted heteroarylcarbonyl N-heteroarylamino, optionally substituted pyrimidinyl-N-arylamino, substituted or unsubstituted Aryl carbonyl N-alkylamino, optionally substituted pyrimidinyl-N-heteroarylamino, optionally substituted heteroarylcarbonyl N-alkylamino, alkoxycarbonylamino, carbonylaminoalkyl alkenyloxy, alkynyloxy carbonylaminoalkyl, cycloalkoxycarbonyl Amino, cycloalkylalkoxycarbonyl Amino, carbonylaminoalkyl ;b alkenyloxy, alkynyloxy ;b carbonylaminoalkyl, aryloxycarbonylamino, alkoxycarbonyl Amino Aryl, Aryl carbonyl Amino alkyenyloxy, Arylalkinyoxycarbonylamino, heteroaryloxycarbonyl Amino, heteroarylalkoxycarbonyl Amino, Heteroaryl carbonylaminoalkyl alkyenyloxy, Heteroarylalkinyoxycarbonylamino, heterocyclyloxycarbonyl Amino, heterocyclylalkoxycarbonyl Amino, Heterocyclyl carbonylaminoalkyl alkyenyloxy, Heterocyclylalkinyoxycarbonylamino, alkoxycarbonyl N-alkylamino, alkenyloxycarbonyl-N-alkylamino, Alkynyloxycarbonyl-N-alkylamino, cycloalkoxycarbonyl-N-alkylamino, cycloalkylalkoxycarbonyl-N-alkylamino, Cycloalkylalkenyloxycarbonyl-N-alkylamino, Cycloalkylalkinyloxycarbonyl-N-alkylamino, aryloxycarbonyl N-alkylamino, arylalkoxycarbonyl-N-alkylamino, Arylalkenyloxycarbonyl-N-alkylamino, Arylalkinyoxycarbonyl-N-alkylamino, heteroarylalkoxycarbonyl-N-alkylamino, Heteroarylalkenyloxycarbonyl-N-alkylamino, Heteroarylalkinyloxycarbonyl-N-alkylamino, heterocyclylalkoxyzarbonyl-N-alkylamino, Heterocyclylalkenyloxycarbonyl-N-alkylamino, Heterocyclylalkinyoxycarbonyl-N-Alkyl Amino, Formyl, halo, haloalkyl, haloalkenyl, haloalkynyl, haloalkoxy, haloalkenyloxy, alkynyloxy Halogen, Thio, halo alkenylthio, alkynylthio Halogen, haloalkylamino, haloalkenyl Amino, alkynyl-Halogen, haloalkylsulfonyl, halo alkenylsulphonyl, alkynylsulfonyl Halogen, haloalkylsulphinyl, Halogen alkenylsulfinyl, alkynylsulfinyl Halogen, haloalkylcarbonyl, acyl halide, alkynylcarbonyl Halogen, haloalkoxy carbonyl, haloalkenyloxy carbonyl, Halogen alkynyloxy carbonyl, carbonyl haloalkylamino, alkylsulfonylaminocarbonyl haloalkenyl, alkynyl-carbonyl halide, halo alkoxycarbonylamino, haloalkenyloxy carbonylaminoalkyl, carbonylaminoalkyl alkynyloxy Halogen, alkoxyalkoxy, arylalkoxy Alkoxy, Cyano, nitro, or a radical selected from the group consisting of Alkyl-nh-N=CH-, Aryl - (CH2) n nh N=CH-, Alkoxy N=CH-, Aryl - (CH2) n ═CH-O-N-, Alkyl-nh-Co - and arylalkyl nh-Co - and R5 optionally Mono - or polysubstituted, by identical or different Alkyl, Alkenyl, alkynyl, Cycloalkyl, Cycloalkenyl, cycloalkylalkyl, Cycloalkyl Alkenyl, cycloalkylalkynyl, Aryl, aralkyl, aralkenyl, arylalkynyl, Heteroaryl, heteroarylalkyl, heteroarylalkenyl, heteroarylalkynyl, Heterocyclyl, heterocyclylalkyl, heterocyclylalkylenyl, heterocyclylalkynyl, Hydroxy, Alkoxy, alkenyloxy, alkynyloxy, Cycloalkoxy, cycloalkylalkoxy, cvcloalkvl alkenyloxy, alkynyloxy cvcloalkvl, cycloalkenyloxy, aryloxy, arylalkoxy, Aryl sulfonyloxy, Aryl alkynyloxy, heteroaryloxy, heteroarylalkoxy, Heteroaryl alkenyloxy, alkynyloxy Heteroaryl, heterocyclyloxy, heterocyclylalkoxy, Heterocyclyl alkenyloxy, alkynyl Heterocyclyl-oxy, Thio, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, ;b alkylthio, alkenylthio ;b, cycloalkylalkynyl Thio, cyclo alkenylthio, arylthio, arylalkylthio, arylalkenyl Thio, Aryl alkynylthio, heteroarylthio, Heteroaryl alkylthio, alkenylthio Heteroaryl, heteroarytatkynyt Thio, heterocyclic Thio, heterocyclic alkylthio, alkenylthio Heterocyclyl, heterocyclylalkynyl Thio, Amino, optionally substituted Mono - or Dialkylamino, optionally substituted Mono - or Diarylamino, optionally substituted Mono - or Di-heteroarylamino, optionally substituted N-Alkyl-N-arylamino, optionally substituted N-Alkyl-N-heteroarylamino, alkenylamino, alkynylamino, cycloalylamin, cycloalkenylamino, Heterocyclyl alkylamino, heterocyclylalkylenyl Amino, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, cycloalkylalkylsulfonyl, alkenylsulphonyl ;b, cycloalkylalkynyl sulfonyl, Aryl sulfonyl, Aryl sulfonyl, Aryl alkenylsulphonyl, arylalkynyl sulfonyl, heteroarylsulfonyl, Heteroaryl Alkyl sulfonyl, Heteroaryl alkenylsulphonyl, heteroarytatkynyt sulfonyl, heterocyclylsulphonyl, heterocyclylaminocarbonyl, alkenylsulphonyl Heterocyclyl, heterocyclylalkynyl sulfonyl, sulfinyl, alkenylsulfinyl, alkynylsulfinyl, cyclo Alkyl sulfinyl, ;b alkylsulfinyl, alkenylsulfinyl cvcloalkvl, alkynylsulfinyl cvcloalkvl, arylsulfinyl, Aryl Alkyl sulfinyl, Aryl alkenylsulfinyl, alkynylsulfinyl Aryl, hetero arylsulfinyl, alkylsulfinyl Heteroaryl, heteroarylalkenyl sulfinyl, phenylsulfinyl heteroarytatkynyt, Heterocyclyl sulfinyl, Aryl Alkyl sulfinyl, phenylsulfinyl heterocyclylalkylenyl, Heterocyclyl alkynylsulfinyl, aminosulfonyl, optionally substituted Mono - or dialkylaminosulfonyl, aminosulfonyl optionally substituted Mono - or Di, optionally substituted Mono - or Di-heteroarylaminosulfonyl are, optionally substituted N-Alkyl-N- arylaminosulfonyl, N-Alkyl-N-heteroarylaminosulfonyl are optionally substituted, alkylsulfonyloxy, phenylsulfonyloxy Alkenyl, alkynyl sulfonyloxy, cyclo Alkyl sulfonyloxy, alkylsulfonyloxy ;b, sulfonyloxy ;b Alkenyl, alkynyl sulfonyloxy cvcloalkvl, arylsulfonyloxy, alkylsulfonyloxy Aryl, aralkyl sulfonyloxy, Aryl sulfonyloxy alkynyl, Heteroaryl sulfonyloxy, alkylsulfonyloxy Heteroaryl, heteroarylalkenyl sulfonyloxy, phenylsulfonyloxy heteroarytatkynyt, sulfonyloxy Heterocyclyl, heterocyclylalkyl sulfonyloxy, phenylsulfonyloxy heterocyclylalkylenyl, sulfonyloxy heterocyclylalkynyl, aryloxycarbonylsmino, alkenylsulphonyl Amino, sulfonylamino alkynyl, Cycloalkyl sulfonyl Amino, Amino Alkyl sulfonic ;b, ;b alkenylsulphonyl Amino, cycloalkylalkynyl sulfonylamino, arylsulfonylamino, isopropylsulfonylamino Aryl, arylalkenyl sulfono-Amino, sulfonylamino arylalkynyl, heteroarylsulfonyl Amino, Heteroaryl isopropylsulfonylamino, heteroarylalkenyl sulfono-Amino, sulfonylamino heteroarytatkynyt, alkylsulfonyl N-alkylamino, alkenylsulphonyl-N-alkylamino, N-Alkyl alkynylsulfonyl-N-alkylamino, cycloalkylsulfonyl-N-alkylamino, cylcoalkylalkylsulfonyl-N-alkylamino, Cycloalkylalkenylsulfonyl-N-alkylamino, Cycloalkylalkinylsulfonyl-N-alkylamino, arylsulfonyl N-alkylamino, heteroarylsulfonyl-N-alkylamino, Arylalkylsulfonyl-N-alkylamino, Heteroarylalkylsulfonyl-N-alkylamino, Arylalkenylsulfonyl-N-alkylamino, Heteroarylalkenylsulfononyl-N-alkylamino, Arylalkinylsulfonyl-N-alkylamino, Heteroarylalkinylsulfonyl-N-alkylamino, heterocyclylsulfonyl-N-alkylamino, heterocyclylalkylsulfonyl-N-alkylamino, Heterocyclylalkenylsulfonyl-N-alkylamino, Heterocyclylalkinylsulfonyl-N-alkylamino, carbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, alkylcarbonylaminoalkyl ;b, alkenylcarbonyl ;b, cycloalkylalkynyl carbonyl, Aryl carbonyl, Aryl Alkyl carbonyl, alkenylcarbonyl Aryl, arylalkynyl carbonyl, heteroarylcarbonyl, heteroarylalkylcarbonyl, heteroarylalkenyl, heteroarytatkynyt carbonyl, heterocyclylcarbonyl, heterocyclylalkylcarbonyl, heterocyclylalkylenyl, heterocyclylalkynyl carbonyl, Carboxyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkoxycarbonyl, cycloalkylalkoxycarbonyl, Cycloalkyl-lower alkenyloxy, alkynyloxy Cycloalkyl carbonyl, aryloxycarbonyl, arylalkoxycarbonyl, Aryl carbonyl alkenyloxy, alkynyloxy carbonyl Aryl, heteroaryloxycarbonyl, heteroarylalkoxycarbonyl, Heteroaryl-lower alkenyloxy, alkynyloxy carbonyl Heteroaryl, heterocyclyloxycarbonyl, heterocyclylalkoxycarbonyl, alkenyloxycarbonyl Heterocyclyl, Heterocyclyl alkynyloxy carbonyl, Amino carbonyl, optionally substituted Mono - or dialkylaminocarbonyl, optionally substituted Mono - or diarylaminocarbonyl, optionally substituted Mono - or Di- Heteroarylaminocarbonyl, optionally substituted N-Alkyl-N- arylaminocarbonyl, optionally substituted N-Alkyl-N- Heteroarylaminocarbonyl, optionally substituted alkylcarbonylamino, substituted or unsubstituted alkylcarbonyl-N-Alkyl Amino, substituted or unsubstituted arylcarbonylamino, substituted or unsubstituted Aryl carbonyl N-arylamino, Amino optionally substituted Heteroaryl, optionally substituted heteroarylcarbonyl N-heteroarylamino, optionally substituted pyrimidinyl-N-arylamino, substituted or unsubstituted Aryl carbonyl N-alkylamino, optionally substituted pyrimidinyl-N-heteroarylamino, optionally substituted heteroarylcarbonyl N-alkylamino, alkoxycarbonylamino, carbonylaminoalkyl alkenyloxy, alkynyloxy carbonylaminoalkyl, cycloalkoxycarbonyl Amino, cycloalkylalkoxycarbonyl Amino, carbonylaminoalkyl ;b alkenyloxy, alkynyloxy ;b carbonylaminoalkyl, aryloxycarbonylamino, alkoxycarbonyl Amino Aryl, Aryl carbonyl Amino alkyenyloxy, Arylalkinyoxycarbonylamino, heteroaryloxycarbonyl Amino, heteroarylalkoxycarbonyl Amino, Heteroaryl carbonylaminoalkyl alkyenyloxy, Heteroarylalkinyoxycarbonylamino, heterocyclyloxycarbonyl Amino, heterocyclylalkoxycarbonyl Amino, Heterocyclyl carbonylaminoalkyl alkyenyloxy, Heterocyclylalkinyoxycarbonylamino, alkoxycarbonyl N-alkylamino, alkenyloxycarbonyl-N-alkylamino, Alkynyloxycarbonyl-N-alkylamino, cycloalkoxycarbonyl-N-alkylamino, cycloalkylalkoxycarbonyl-N-alkylamino, Cycloalkylalkenyloxycarbonyl-N-alkylamino, Cycloalkylalkinyloxycarbonyl-N-alkylamino, aryloxycarbonyl N-alkylamino, arylalkoxycarbonyl-N-alkylamino, Arylalkenyloxycarbonyl-N-alkylamino, Arylalkinyoxycarbonyl-N-alkylamino, heteroarylalkoxycarbonyl-N-alkylamino, Heteroarylalkenyloxycarbonyl-N-alkylamino, Heteroarylalkinyoxycarbonyl-N-alkylamino, heterocyclylalkoxyzarbonyl-N-alkylamino, Heterocyclylalkenyloxycarbonyl-N-alkylamino, Heterocyclylalkinyoxycarbonyl-N-Alkyl Amino, Formyl, halo, haloalkyl, haloalkenyl, haloalkynyl, haloalkoxy, haloalkenyloxy, alkynyloxy Halogen, Thio, halo alkenylthio, alkynylthio Halogen, haloalkylamino, haloalkenyl Amino, Halogen alkynylamino, haloalkylsulfonyl, halo alkenylsulphonyl, alkynylsulfonyl Halogen, haloalkylsulphinyl, Halogen alkenylsulfinyl, alkynylsulfinyl Halogen, haloalkylcarbonyl, acyl halide, alkynylcarbonyl Halogen, haloalkoxy carbonyl, haloalkenyloxy carbonyl, Halogen alkynyloxy carbonyl, carbonyl haloalkylamino, alkylsulfonylaminocarbonyl haloalkenyl, alkynyl-carbonyl halide, halo alkoxycarbonylamino, haloalkenyloxy carbonylaminoalkyl, carbonylaminoalkyl alkynyloxy Halogen, alkoxyalkoxy, arylalkoxy Alkoxy, Cyano, nitro, or a radical selected from the group consisting of Alkyl-nh-N=CH-, Aryl - (CH2) n nh N=CH-, Alkoxy N=CH-, Aryl (CH2) n ═CH-O-N-, Alkyl-nh-Co - and Aryl-Alkyl-nh-Co -, substituted Heteroaryl, Heterocyclyl or Aryl.  3. Benzoyl derivatives according to claim 1 or 2, wherein R1, R2, R3 independently hydrogen, Halogen, nitro, cyano, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylsulfonyloxy, alkylsulfonylamino, alkylsulfonyl N-alkylamino, Phenyl, benzyl, wherein the latter groups substituted with one or more thirteen, identical or different substituents selected from the group consisting of Halogen, nitro, cyano, alkyl, halo, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkoxy and alkylthio substituted; R4 hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl, the latter four groups are optionally substituted by one or more, identical or different substituents selected from the group consisting of Halogen, nitro, cyano, alkyl, cycloalkyl, alkenyl, alkoxy, alkylthio substituted; R5 optionally mono - or polysubstituted, by identical or different Halogen, nitro, cyano, Formyl, amino, Phenyl, benzyl, (C1 -C6) alkyl, (C2 -C6) alkenyl, (C2 -C6) alkynyl, (C3 -C8) cycloalkyl, (C1 -C6) alkoxy, (C1 -C6) alkylamino, Di (C1 -C6) alkylamino, (C1 -C6) alkoxycarbonyl, (C1 -C6) alkylaminocarbonyl, Di (C1 -C6) - alkylaminocarbonyl, (C1 -C6) alkanoyl, (C1 -C6) alkylcarbonylamino, (C1 -C6) - alkylcarbonyl (C1 -C6) alkylamino, (C1 -C6) - carbonyl-Di - (C1 -C6) alkylamino, (C1 -C6) alkylthio, (C1 -C6) alkylsulfinyl, (C1 -C6) alkylsulphonyl, (C1 -C6) cycloalkyl, (C1 -C6) alkylsulfonyl - (C1 -C6) alkylamino, (C1 -C6) alkylsulphonyl Di (C1 -C6) alkyl amino, the latter groups substituted with one or more 22 identical or different substituents selected from the group consisting of Halogen, nitro, cyano, (C1 -C6) alkyl, (C3 -C6) cycloalkyl, (C2 -C6) alkenyl, (C2 -C6) alkynyl, (C1 -C6) alkoxy, (C1 -C6) alkylthio or three to six membered, saturated, partially saturated or unsaturated heterocycle, up to four heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur atom may, substituted, substituted Phenyl, or three to six-membered, saturated, partially saturated or unsaturated heterocyclic group, up to four heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur atom may; A from A divalent moiety S, so, so2, and noa ; B A saturated or A double bond-containing one or two carbon atoms and from existing chain, optionally substituted with alkyl, halo, alkoxy or substituted aryl; E is A bond, crc Rd, noc, S, so, so2, O and co; R6 (C1 -C6) alkylthio, (C1 -C6) alkylsulfinyl, (C1 -C6) alkylsulfonyl, cyano, cyanato, Thiocyanato, Halogen or orf ; A divalent moiety selected from the group O Y, S, N-(C1 -C6) alkyl or chr7 ; R7 hydrogen, (C1 -C6) alkyl, (C3 -C8) cycloalkyl, (C1 -C6) alkoxy, (C1 -C6) alkoxy (C1 -C6) alkyl, (C1 -C6) alkanoyl, (C1 -C6) alkoxycarbonyl, (C1 -C6) alkylthio, Phenyl, wherein the hydrocarbon radicals substituted with one or more portion of the eight last, identical or different substituents selected from the group consisting of Halogen, (C1 -C3) alkylthio and (C1 -C3) alkyloxy substituted; Z is A bond, ch2 or chr7 ; R8 hydrogen, (C1 -C6) alkyl or (C1 -C6) alkoxycarbonyl; R9 hydrogen, (C1 -C6) alkyl, (C3 -C8) - cycloalkyl or halo (C1 -C6) alkyl; R10 hydrogen, (C1 -C6) alkyl, (C2 -C6) alkenyl, (C1 -C6) alkynyl, (C3 -C8) cycloalkyl, Phenyl, benzyl, wherein the six groups are optionally substituted by one or more last-mentioned radicals, identical or different substituents selected from the group consisting of Halogen, cyano, nitro and (C1 -C6) alkoxy; R11 hydrogen, Formyl, (C1 -C6) alkyl, halo (C1 -C6) alkyl, (C1 -C6) alkoxy (C1 -C6) alkyl or A group L-R12 ; A divalent moiety selected from the group so L2, co and chrg co; R12 (C1 -C6) alkyl, halo (C1 -C6) alkyl, unsubstituted or substituted by one or more, identical or different substituents selected from the group consisting of cyano, nitro, (C1 -C3) alkyl, (C1 -C3) alkoxy, halo (C1 -C3) alkyl and halo (C1 -C3) alkoxy substituted Phenyl; Ra hydrogen, Halogen, cyano, nitro, Formyl, (C1 -C6) alkyl, (C3 -C6) cycloalkyl, (C2 -C6) alkenyl, (C2 -C6) alkynyl, (C1 -C6) alkanoyl and (C1 -C6) alkylsulfonyl, wherein the hydrocarbon portion of the six lastmentioned groups optionally with one or more, identical or different substituents selected from the group consisting of Halogen, nitro, cyano, (C1 -C6) alkyl, (C3 -C8) cycloalkyl, (C2 -C6) alkenyl, (C2 -C6) alkynyl, (C1 -C6) alkoxy and (C1 -C6) substituted alkylthio; Rc and Rd independently hydrogen, Halogen, nitro, cyano, (C1 -C6) alkyl, halo (C1 -C6) alkyl, (C3 -C8) cycloalkyl, (C2 -C6) alkenyl, halo (C2 -C6) alkenyl, (C2 -C6) alkynyl, halo (C2 -C6) alkynyl, (C1 -C6) alkoxy, halo (C1 C6) alkoxy, (C1 -C6) alkylthio, halo (C1 C6) - alkylthio, (C1 -C6) alkanoyl, halo (C1 -C6) alkylsulfonyl, (C1 -C6) alkoxycarbonyl, halo (C1 -C6) alkoxycarbonyl, aminocarbonyl, (C1 -C6) alkanoyl and (C1 -C6) alkylsulfonyl; Re hydrogen, Formyl, (C1 -C6) alkyl, (C3 -C8) cycloalkyl, (C2 -C6) alkenyl, (C2 -C6) alkynyl, (C1 -C6) alkanoyl and (C1 -C6) alkylsulfonyl, wherein the hydrocarbon portion of the six lastmentioned radicals substituted with one or more, identical or different substituents selected from the group consisting of Halogen, nitro, cyano, (C1 -C6) alkyl, cycloalkyl, (C2 -C6) alkenyl, (C2 -C6) - (C1 -C6) alkynyl, (C1 -C6) alkoxy and (C1 -C6) may be substituted alkylthio; Rf hydrogen, (C1 -C6) alkyl, halo (C1 -C6) alkyl, (C1 -C6) alkanoyl, (C1 -C6) alkoxycarbonyl, (C1 -C6) alkylsulfonyl, Halogen (C1 -C6) alkylsulfonyl, benzoyl or Phenylsufonyl, wherein the concentration of the latter two groups optionally substituted by one or more, identical or different substituents selected from the group (C1 -C6) alkyl, halo (C1 -C6) alkyl, (C1 -C6) alkoxy, halo (C1 -C6) alkoxy, Halogen, cyano and nitro substituted; Rg and Rh independently hydrogen or (C1 -C6) alkyl, and w 0, 1, 2 or 3 are.  4. Benzoyl derivatives according to any one of claims 1 to 3, wherein R1, R2, R3 independently hydrogen, Halogen, nitro, cyano, (C1 -C6) alkyl, (C3 -C8) cycloalkyl, (C2 -C6) alkenyl, (C2 -C6) alkynyl, (C1 -C6) alkoxy, (C1 -C6) alkylthio, (C1 -C6) radical, (C1 -C6) alkylsulphonyl, (C1 -C6) alkylsulfonyloxy, (C1 -C6) cycloalkyl, (C1 -C6) alkylsulfonyl-N-(C1 -C6) alkyl amino, Phenyl, benzyl, substituted by one or more groups of the latter with the thirteen, identical or different substituents selected from the group consisting of Halogen, nitro, cyano, (C1 -C3) alkyl, halo (C1 -C3) alkyl, cyclopropyl, (C2 -C4) alkenyl, (C2 -C4) alkynyl, (C1 -C3) alkoxy, halo (C1 -C3) alkoxy and alkylthio substituted; R4 (C1 -C4) alkyl, hydrogen, cyano, (C2 -C4) alkenyl, (C2 -C4) alkynyl, (C3 -C6) - cycloalkyl, the latter three groups are optionally substituted by one or more, identical or different substituents selected from the group consisting of Halogen, cyano, (C1 -C3) alkoxy, (C1 -C3) substituted alkoxy, optionally substituted by one or more and the former, identical or different substituents selected from the group consisting of Halogen, cyano, (C3 -C6) cycloalkyl, (C1 -C3) alkoxy, (C1 -C3) substituted alkylthio; R5 optionally mono - or polysubstituted, the same or different Halogen, nitro, cyano, Formyl, amino, Phenyl, benzyl, (C1 -C4) alkyl, (C2 -C4) alkenyl, (C2 -C4) alkynyl, (C3 -C6) cycloalkyl, (C1 -C4) alkoxy, (C1 -C4) alkylamino, Di (C1 -C4) alkylamino, (C1 -C4) alkoxycarbonyl, (C1 -C4) alkylaminocarbonyl, Di (C1 -C4) - alkylaminocarbonyl, (C1 -C4) alkanoyl, (C1 -C4) alkoxy, (C1 -C4) alkylthio, (C1 -C4) alkylsulfinyl, (C1 -C4) alkylsulfonyl, substituted Phenyl, or three to six-membered, saturated, partially saturated or unsaturated heterocyclic group, up to four heteroatoms selected from nitrogen, oxygen and sulfur atom may; A from A divalent moiety S, so, and so2 ; and B A saturated or A double bond-containing one or two carbon atoms existing chain, optionally substituted with one or two identical or different substituents selected from the group (C1 -C3) alkyl, halo (C1 -C3) alkyl, (C1 -C3) alkoxy or Halogen (C1 -C3) is substituted; E is A bond, crc Rd, so2 and co; R6 (C1 -C3) alkylthio, (C1 -C3) alkylsulfonyl, cyano, cyanato, Thiocyanato, Halogen or orf ; Y A divalent moiety selected from the group O or chr7 ; R7 hydrogen, (C1 -C6) alkyl, (C3 -C8) cycloalkyl, (C1 -C6) alkoxy (C1 -C6) alkyl, (C1 -C5) alkanoyl, (C1 -C6) alkoxycarbonyl, Phenyl, optionally substituted by one or more said six lastmentioned radicals, are identical or different Halogen atoms; R9 (C1 -C6) alkyl, (C3 -C6) - cyc(...)
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(DE19840337) LEGAL DETAILS FOR DE19840337  Actual or expected expiration date=2001-10-11    Legal state=DEAD    Status=LAPSED     Event publication date=1998-09-04  Event code=DE/APP  Event indicator=Pos  Event type=Examination events  Application details  Application country=DE DE19840337  Application date=1998-09-04  Standardized application number=1998DE-1040337     Event publication date=2000-03-09  Event code=DE/A1  Event type=Examination events  Doc. laid open (First publication)  Publication country=DE  Publication number=DE19840337  Publication stage Code=A1  Publication date=2000-03-09  Standardized publication number=DE19840337     Event publication date=2000-05-25  Event code=DE/8127  Event type=Change of name or address  Event type=Reassignment  New person/name/address of the applicant Aenderung in person, namen oder wohnort des anmelders    Event publication date=2001-01-11  Event code=DE/8127  Event type=Change of name or address  Event type=Reassignment  New person/name/address of the applicant Aenderung in person, namen oder wohnort des anmelders    Event publication date=2001-10-11  Event code=DE/8139  Event indicator=Neg  Event type=Event indicating Not In Force  Disposal/non-payment of the annual fee Erledigt wegen nichtz. d. jahresgeb.
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