(ES-477353) intensity of the infection according to the indices of an evaluation scale that va of 100 (it plants healthy) to Or (it plants complete infected mind). EXAMPLE 23. 5. Determination of the fitotoxicidad The leaves were grapevine plant CB. Dolcetto, cultivated in flowerpot in an atmosphere equipped to 25QC and 60% of relative moist soil, sprinkling its two faces with the products that try on in a hidroacetonica solution 10. To 20% do acetone (bowl. /vol.). After 7 days the gravity of the phytotoxic symptoms was evaluated do forms line of vision according to indices of one associates of evaluation that va of damaged) to Or (it plants healthy). 15. = 1 CLAIMS Described to the object of the present invento' “the following claims would sedeclaran new and of own invention. 20. 1. A procedure for the preparation do new acyl-anilines of activity fungicide, the general formula X - (CH 2) r. 1. C //R R where 100 (plant totally 32. R and R 1 (different equals or to each other) = H; CH 3; 3. R and R 4 (different equals or to each other) = H; alkyl C 1 - C 3; 5. or together 3 R and R 4 is (CH 2 =) X = - C-R 9; - C-0-R 9 (R 9 CA n l or. or or (R 5 = alkyl or alquilideno); alkyl) 15. N = 0,1 Z = phenyl optionally replaced; - (CH) - AND; CH 9 - C-R 8 and R 2 = H, CH 3; m = 1,2; And = alquinilo C 2 - Cs 8; cicloalquilo C 3 - Cs 8; piridilo; heterocyclic groups containing 2 or 3 have to you roatomos, one of them different one from nitrogen; R 8 5: CH 3; alcoximetilo; halometilo; 0-alkyl, characterized because do is made react an aniline the general formula: 25. S1/R4 S 1/R4 C X - (CH 2) n,/ R 2. CS H 5; n. 3 CS H 7; - CH 2 - CH= =CH 2; - CH=CH-CH 3; halometilo; CL; F; CNN; Or-Alkyl; S-Alkyl; alcoximetilo; = alkyl C 1 - C 3); CNN; - CH. (OR 5) 2 rt /7 CNN (R 6 and R 7 = H, or \ 7 Or R or phenyl n optionally replaced; fenil-acetyl, furilo; tienilo; NH (where R, R 1, R 3, R 4, indicated) in a dimetilformamida inert dissolvent and in the presence of or of a base would accept of halogenhldrico acid, with clo- 5. ruro of a carboxylic acid of the formula: CL (where Z has the indicated meaning before). 2. A procedure according to the claim 10. 1, characterized in a variant do its accomplishment, because when in the general formula Z it means - CH 2 - 00-CH 3, it makes react, on an inert dissolvent, the aniline d9 the formula: R 3 15. X - (CH 2); ' (in giving R, R 1, R 3, R 4, on claim 1) 20. with dicetono CH 2 3. A procedure for the preparation do new acyl-anilines do activity fungicide. 25. According To under I describe and vindicates in the present descriptive memory that consists of 33 pages in leaf and written to machine by a single do his Xs and n have the meaning before C Z (III) Or , R 4 NH Xs and n have the set out meaning = Or H 2 -/'= OR faces. - 34 You Hoist you go i to 1 FEBRUARY, 1979 Pea. JAtM P. P. Finnolz PIEBALD JESUS
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