A PROCEDURE FOR THE PREPARATION OF NEW ACIL-ANILINASDE ACTIVITY FUNGICIDES. 机翻标题: 暂无翻译,请尝试点击翻译按钮。

源语言标题
(ES-477353) Un procedimiento para la preparacion de nuevas acil-anilinasde actividad fungicidas.
公开号/公开日
ES477353 A1 1980-01-16 [ES-477353] / 1980-01-16
申请号/申请日
1979ES-0477353 / 1979-02-01
发明人
;
申请人
MONTEDISON;
主分类号
IPC分类号
A01N-033/06A01N-037/22A01N-037/30A01N-037/42A01N-037/46A01N-043/06A01N-043/08A01N-043/10A01N-043/40A01N-053/12C07C-067/00C07C-231/02C07C-233/18C07C-233/31C07C-233/47C07C-233/53C07C-233/58C07C-233/73C07C-233/88C07C-235/56C07C-235/68C07C-235/80C07C-237/22C07C-253/00C07C-255/29C07C-313/00C07C-323/41C07C-323/42C07C-323/59C07C-323/60C07D-307/54C07D-333/22C07D-333/24
摘要
(ES-477353) Acyl anilines are disclosed having the formula <IMAGE> (I) wherein R and R1 (like or unlike each other)=H; CH3; C2H5; n.C3H7; -CH2-CH=CH2; -CH=CH-CH3; R3 and R4 (like or unlike each other)=H; alkyl C1-C3; halomethyl; Cl; F; CN; O-alkyl; S-alkyl; alkoxymethyl; or R3 and R4 together are (CH2=) <IMAGE> (R9=alkyl C1-C3); CN; -CH(OR5)2 (R5=alkyl or alkylidene ); <IMAGE> (R6 and R7=H, alkyl) 'n=0,1 Z=phenyl optionally substituted; <IMAGE> And R2=H, CH3; m=1,2; Y=alkynyl C2-C8; phenyl optionally substituted; phenyl-acetyl; furyl, thienyl; pyridyl; heterocyclic groups containing 2 or 3 heteroatoms, one of them different from nitrogen; R8=CH3; alkoxymethyl; halomethy; O-alkyl.  The compounds of formula I are endowed with a high fungicidal activity and with a low phytotoxicity.  (From US4291049 A)
机翻摘要
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地址
代理人
代理机构
;
优先权号
1978IT-0019896 1978-02-02 1978IT-0025295 1978-07-04
主权利要求
(ES-477353) intensity of the infection according to the indices of an evaluation scale that va of 100 (it plants healthy) to Or (it plants complete infected mind). EXAMPLE 23. 5. Determination of the fitotoxicidad The leaves were grapevine plant CB. Dolcetto, cultivated in flowerpot in an atmosphere equipped to 25QC and 60% of relative moist soil, sprinkling its two faces with the products that try on in a hidroacetonica solution 10. To 20% do acetone (bowl. /vol.). After 7 days the gravity of the phytotoxic symptoms was evaluated do forms line of vision according to indices of one associates of evaluation that va of damaged) to Or (it plants healthy). 15. = 1 CLAIMS Described to the object of the present invento' “the following claims would sedeclaran new and of own invention. 20. 1. A procedure for the preparation do new acyl-anilines of activity fungicide, the general formula X - (CH 2) r. 1. C //R R where 100 (plant totally 32. R and R 1 (different equals or to each other) = H; CH 3; 3. R and R 4 (different equals or to each other) = H; alkyl C 1 - C 3; 5. or together 3 R and R 4 is (CH 2 =) X = - C-R 9; - C-0-R 9 (R 9 CA n l or. or or (R 5 = alkyl or alquilideno); alkyl) 15. N = 0,1 Z = phenyl optionally replaced; - (CH) - AND; CH 9 - C-R 8 and R 2 = H, CH 3; m = 1,2; And = alquinilo C 2 - Cs 8; cicloalquilo C 3 - Cs 8; piridilo; heterocyclic groups containing 2 or 3 have to you roatomos, one of them different one from nitrogen; R 8 5: CH 3; alcoximetilo; halometilo; 0-alkyl, characterized because do is made react an aniline the general formula: 25. S1/R4 S 1/R4 C X - (CH 2) n,/ R 2. CS H 5; n. 3 CS H 7; - CH 2 - CH= =CH 2; - CH=CH-CH 3; halometilo; CL; F; CNN; Or-Alkyl; S-Alkyl; alcoximetilo; = alkyl C 1 - C 3); CNN; - CH. (OR 5) 2 rt /7 CNN (R 6 and R 7 = H, or \ 7 Or R or phenyl n optionally replaced; fenil-acetyl, furilo; tienilo; NH (where R, R 1, R 3, R 4, indicated) in a dimetilformamida inert dissolvent and in the presence of or of a base would accept of halogenhldrico acid, with clo- 5. ruro of a carboxylic acid of the formula: CL (where Z has the indicated meaning before). 2. A procedure according to the claim 10. 1, characterized in a variant do its accomplishment, because when in the general formula Z it means - CH 2 - 00-CH 3, it makes react, on an inert dissolvent, the aniline d9 the formula: R 3 15. X - (CH 2); ' (in giving R, R 1, R 3, R 4, on claim 1) 20. with dicetono CH 2 3. A procedure for the preparation do new acyl-anilines do activity fungicide. 25. According To under I describe and vindicates in the present descriptive memory that consists of 33 pages in leaf and written to machine by a single do his Xs and n have the meaning before C Z (III) Or , R 4 NH Xs and n have the set out meaning = Or H 2 -/'= OR faces. - 34 You Hoist you go i to 1 FEBRUARY, 1979 Pea. JAtM P. P. Finnolz PIEBALD JESUS
法律状态
(ES-477353) LEGAL DETAILS FOR ES477353  Actual or expected expiration date=1999-02-01    Legal state=DEAD    Status=EXPIRED     Event publication date=1979-02-01  Event code=ES/APP  Event indicator=Pos  Event type=Examination events  Application details  Application country=ES ES477353  Application date=1979-02-01  Standardized application number=1979ES-0477353     Event publication date=1980-01-16  Event code=ES/A1  Event indicator=Pos  Event type=Event indicating In Force  Patent of invention  Publication country=ES  Publication number=ES477353  Publication stage Code=A1  Publication date=1980-01-16  Standardized publication number=ES-477353     Event publication date=1999-02-01  Event code=ES/EEDX  Event indicator=Neg  Event type=Event indicating Not In Force  Patent has expired
专利类型码
A1
国别省市代码
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