Substituted n-propargyl anilines, process for their preparation and their use as fungicides 机翻标题: 暂无翻译,请尝试点击翻译按钮。

公开号/公开日
EP0010673 A2 1980-05-14 [EP--10673]EP0010673 A3 1980-07-23 [EP--10673]EP0010673 B1 1982-01-27 [EP--10673] / 1980-05-141980-07-231982-01-27
申请号/申请日
1979EP-0103965 / 1979-10-15
发明人
STETTER, JORG, DR.;LUNKENHEIMER, WINFRIED, DR.;BRANDES, WILHELM, DR.;
申请人
BAYER;
主分类号
IPC分类号
A01N-037/22A01N-037/26A01N-037/34A01N-043/08A01N-043/653A01N-043/80A01N-047/20A01N-047/48C07C-067/00C07C-233/07C07C-233/09C07C-233/13C07C-233/88C07C-235/16C07C-235/68C07C-239/00C07C-253/00C07C-255/27C07C-271/28C07C-301/00C07C-303/28C0
摘要
(EP--10673) 1.  Substituted N-propargyl-anilines of the general formula see diagramm : EP0010673,P37,F3 in which R**1 , R**2 , R**3 , R**4 and R**5 represent hydrogen and alkyl with 1 to 4 carbon atoms, and furthermore R**1 additionally represents halogen and R**5 additionally represents phenyl which is optionally substituted by halogen, alkyl with 1 to 4 carbon atoms and nitro, and halogen, R**6 represents tetrahydrofuryl, thiophenyl, tetrahydrothiophenyl, optionally methyl- or ethyl-substituted isoxazolyl, and optionally cyano- or thiocyano-substituted alkyl with 1 to 4 and alkenyl and alkinyl each with 2 to 4 carbon atoms, and represents the groupings -CH2 -Az, -CH2 -OR**8 , -CH2 -SR**7 , -OR**7 , -CH2 -OSO2 R**8 , -COOR**7 and see diagramm : EP0010673,P38,F1 wherein R**7 and R**8 represent halogen-, cyano and thiocyano-substituted alkyl with 1 to 4 carbon atoms and alkenyl and alkinyl, with in each case 2 to 4 carbon atoms, which are optionally substituted by the indicated alkyl substituents and represents alkoxyalkyl with 1 to 4 carbon atoms in each alkyl part, and furthermore R**7 can additionally represent unsubstituted alkyl with 1 to 4 carbon atoms, and Az represents pyrazol-1-yl) 1,2,4-triazol-1-yl and imidazol-1-yl.
机翻摘要
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地址
代理人
代理机构
;
优先权号
1978DE-2847287 1978-10-31 1979DE-2927461 1979-07-06
主权利要求
(EP--10673)  1. Substituted One N-Propargyl-aniline the general Forms 1 EMI64.1 in which R1 for Hydrogen, Alkyl or Halogen s.teht, R2 stands for R3 for Hydrogen or Alkyl, for Hydrogen or Alkyl stands, for R4 for Hydrogen or Alkyl stands, R5 fur Hydrogen, Alkyl, Halogen or if necessary substituted Phenyl stands, for R6 for Furyl, Tetrahydrofuryl, Thiophenyl, Tetra hydrothiophenyl;  if necessary by Alkyl substituted Isoxazolyl;  if necessary through Cyano or Thiocyans substituted Alkyl, Alkenyl and Alkinyl;  Dihalogenalkyl;  as well as the Groupings - CH2-Az, -CH2-oR7, -CH2-SR7, - OR7, - SR7, -CH2-OSO2R7, -COOR7 and EMI64.2 stands, how R7 for Alkyl substituted if necessary, Alkenyl, Alkinyl and Alkoxy alkyl stand, and Az for Pyrazol l Yl, 1,2,4-Triazol-l-yl and imidazole l Yl stands. 2. Procedures for the Production of substituted N-Propargyl anilinen, by the fact characterized that one a) N-Propargyl-aniline of the Formula EMI65.1 in which G 1 to R5 the Meaning indicated above have, with Acid Chloride or - bromide and/or - anhydrides of the Formulas EMI65.2 and/or.  EMI65.3 Into which R6 the Meaning indicated above if necessary converts haut, in Presence of a Diluent and in Presence of an Acid Bonding Agent, or b) Anilide of the Formula EMI66.1 in which R1 to R3 and R6 the It interpretation indicated above more haber, with Propargylhalogeniden of the Formula EMI66.2 in which R4 have and R5 the BE interpretation indicated above, and Hal fur Chlorine or Bromine stands, in Presence of an Acid Binder and in Presence of an organic Verdunnungsmittels or in an aqueous-organic Two-phase system in Presence of a Phase Transfer Catalyst converts if necessary;  or individual Connections of the Formula (I), by one c) Halogenacetanilide of the Formula EMI67.1 in which R1bis have R5 the BE interpretation indicated above, and Hai' stands for Chlorine, Bromine or Iodine, with Connections of the Formula B - X (VII) in which X for Az and the Grouping - OR7 or - SR7 stands. and B for Hydrogen or an Alkali Metal stands, if necessary in Presence of a Diluent and in Presence of an Acid Binder converts, or for i) Hydroxyacetanilide Formel if necessary EMI68.1 in which R1 to R5 have the Meaning indicated above, (1) gegebenenalls after Activation mittels Alkali metal with Halides of the Formula Hal - R8 (IX) in which Hal' Bedet indicated above:: tunq has, and R8 for the Rest of R7 as well as the Group -;  Q R7 stands, how R7 those the Meaning indicated above has, in Presence of a Diluent and in Presence of an Acid Binder converts if necessary, or (2) with Dihydropyran of the Formula EMI69.1 in Presence of a Diluent and a given if in Presence of a Catalyst umsetzt1 or e) erfindungsgemasse N-Propargyl-anilide of the Formula EMI69.2 in which G 1 to R4 and R6 the Meaning indicated above have, in actually well-known Way with aqueous Alkalihypohalogenit solutions convert. 3. Fungicides Means, characterized through eznen Content in at least a substituted N-Propargyl aniline in accordance with Anspruc ta v. 4. Procedure for the Fight against Mushrooms, thereby GE marks that one substituted N-Propargyl aniline in accordance with claim 1 on Mushrooms or their lasst. influences Habitat 5. Use of substituted N-Propargyl-aniline in accordance with claim 1 to Bekampfung von Pilzen. 6. Procedures for the Production of fungicides average, thus gekennzeichret, that one substituted N-Fr3- pargyl aniline in accordance with claim 1 with Stretching Means and/or surface-active Means mixes.
法律状态
(EP--10673) LEGAL DETAILS FOR EP0010673  Actual or expected expiration date=1999-10-15    Legal state=DEAD    Status=EXPIRED     Event publication date=1979-10-15  Event code=EP/APP  Event indicator=Pos  Event type=Examination events  Application details  Application country=EP EP79103965  Application date=1979-10-15  Standardized application number=1979EP-0103965     Event publication date=1980-05-14  Event code=EP/A2  Event type=Examination events  Application published without search report  Publication country=EP  Publication number=EP0010673  Publication stage Code=A2  Publication date=1980-05-14  Standardized publication number=EP--10673     Event publication date=1980-05-14  Event code=EP/AK  Event indicator=Pos  Event type=Designated states  Designated contracting states: Benannte vertragsstaaten AT BE CH DE FR GB IT NL SE    Event publication date=1980-05-14  Event code=EP/17P  Event indicator=Pos  Event type=Examination events  Request for examination filed Pruefungsantrag gestellt    Event publication date=1980-07-23  Event code=EP/A3  Event indicator=Pos  Event type=Examination events  Published search report  Publication country=EP  Publication number=EP0010673  Publication stage Code=A3  Publication date=1980-07-23  Standardized publication number=EP--10673     Event publication date=1980-07-23  Event code=EP/AK  Event indicator=Pos  Event type=Designated states  Designated contracting states: Benannte vertragsstaaten AT BE CH DE FR GB IT NL SE    Event publication date=1982-01-27  Event code=EP/B1  Event indicator=Pos  Event type=Event indicating In Force  Patent specification  Publication country=EP  Publication number=EP0010673  Publication stage Code=B1  Publication date=1982-01-27  Standardized publication number=EP--10673     Event publication date=1982-01-27  Event code=EP/AK  Event indicator=Pos  Event type=Designated states  Designated contracting states: Benannte vertragsstaaten AT BE CH DE FR GB IT NL SE    Event publication date=1999-10-15  Event code=EP/EEDX  Event indicator=Neg  Event type=Event indicating Not In Force  Patent has expired MEMBER STATE LEGAL DETAILS FOR AT613  Actual or expected expiration date=1982-10-15    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=AT Corresponding appl: AT79103965  Application date in the designated or member state=1979-10-15   Application number in the designated or member state=1979AT-0103965T Corresponding cc:  Designated or member state=AT Corresponding pat: AT613  Publication stage code in the designated or member state=T  Publication date in the designated or member state=1982-02-15   Publication number in the designated or member state=ATE000613    Event publication date=1982-01-27  Event code=EP/REF  Event type=Entry into national phase  Corresponds to: Corresponding cc:  Designated or member state=AT     Event publication date=1982-10-15  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=AT   Effective date of the event=1982-10-15  MEMBER STATE LEGAL DETAILS FOR BE  Actual or expected expiration date=1982-10-15    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=BE     Event publication date=1982-10-15  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=BE   Effective date of the event=1982-10-15  MEMBER STATE LEGAL DETAILS FOR CH  Actual or expected expiration date=1982-10-31    Legal state=DEAD    Status=EXPIRED   Corresponding cc:  Designated or member state=CH     Event publication date=1982-10-31  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=CH   Effective date of the event=1982-10-31     Event publication date=1983-06-30  Event code=EP/REG  Event code=CH/PL  Event indicator=Neg  Event type=Event indicating Not In Force  Reference to a national code Patent ceased Loeschung/radiation/radiazion Corresponding cc:  Designated or member state=CH  MEMBER STATE LEGAL DETAILS FOR DE  Actual or expected expiration date=1983-07-01    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=DE Corresponding appl: DE2961993    Event publication date=1982-03-11  Event code=EP/REF  Event type=Entry into national phase  Corresponds to: Corresponding cc:  Designated or member state=DE     Event publication date=1983-07-01  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=DE   Effective date of the event=1983-07-01  MEMBER STATE LEGAL DETAILS FOR FR  Actual or expected expiration date=1983-07-29    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=FR     Event publication date=1983-07-29  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=FR   Effective date of the event=1983-07-29  LAPSE BECAUSE OF NON-PAYMENT OF DUE FEES     Event publication date=1983-09-23  Event code=EP/REG  Event code=FR/ST  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Reference to a national code Notification of lapse Constatation de decheances Corresponding cc:  Designated or member state=FR  MEMBER STATE LEGAL DETAILS FOR GB  Actual or expected expiration date=1988-11-18    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=GB     Event publication date=1988-11-18  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=GB   Effective date of the event=1988-11-18  MEMBER STATE LEGAL DETAILS FOR IT  Actual or expected expiration date=1999-10-15    Legal state=DEAD    Status=EXPIRED   Corresponding cc:  Designated or member state=IT     Event publication date=1981-10-06  Event code=EP/ITF  Event indicator=Pos  Event type=Examination events  IT: Translation for a EP patent filed IT: Deposito traduzione di brevetto europeo Corresponding cc:  Designated or member state=IT  MEMBER STATE LEGAL DETAILS FOR NL  Actual or expected expiration date=1983-05-01    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=NL     Event publication date=1983-05-01  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=NL   Effective date of the event=1983-05-01     Event publication date=1983-06-16  Event code=EP/NLV4  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  NL: Lapsed or anulled due to non-payment of the annual fee NL: Vervallen wegens niet betalen van een jaarcijns Corresponding cc:  Designated or member state=NL  MEMBER STATE LEGAL DETAILS FOR SE  Actual or expected expiration date=1985-06-11    Legal state=DEAD    Status=LAPSED   Corresponding cc:  Designated or member state=SE Corresponding appl: SE79103965.4    Event publication date=1982-01-27  Event code=EP/PG25  Event indicator=Neg  Event type=Event indicating Not In Force  Event type=Payment or non-payment notifications  Lapsed in a contracting state announced via postgrant inform. from nat. office to EPO Corresponding cc:  Designated or member state=SE   Effective date of the event=1982-01-27  THE PATENT HAS BEEN ANNULLED BY A DECISION OF A NATIONAL AUTHORITY     Event publication date=1995-01-31  Event code=EP/EUG  Event indicator=Neg  Event type=Event indicating Not In Force  SE: European patent has lapsed SE: Europeiskt patent har upphoert att gaella Corresponding cc:  Designated or member state=SE   Effective date of the event=1985-06-11
专利类型码
A2A3B1
国别省市代码
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