(BR112015020972) Condensed heterocyclic compound, use of condensed heterocyclic composite compound or a salt thereof, method to use an agricultural and horticultural insecticide, method to control pests of agricultural and horticultural insects, the control agent of contagious and insecticide 机翻标题: 暂无翻译,请尝试点击翻译按钮。

源语言标题
(BR112015020972) Condensed heterocyclic compound, use of condensed heterocyclic composite compound or a salt thereof, method to use an agricultural and horticultural insecticide, method to control pests of agricultural and horticultural insects, the control agent of contagious and insecticide
公开号/公开日
BR112015020972 BR112015020972 BR112015020972 / 2019-12-03 2017-07-18 2015-12-15
申请号/申请日
BR112015020972 / 2014-03-14
发明人
AKIYUKI SUWA IKKI YONEMURA KOSUKE FUKATSU TAKASHI FURUYA
申请人
NIHON NOHYAKU
主分类号
IPC分类号
A01N-043/90 A01P-007/04 A61K-031/5025 A61P-033/14 C07D-487/04
摘要
(BR112015020972)
An object of the present invention is to provide and develop novel agricultural and horticultural insecticides in view of the still immense damage caused by insect pests etc. and the emergence of insect pests resistant to existing insecticides in crop production in the fields of agriculture, horticulture and the like. Provided are a condensed heterocyclic compound represented by the general formula (I): {wherein A 1 , A 2 and A 3 may be the same or different, and each represent a nitrogen atom or a CH group, R 1 represents an alkyl group or the like, R 2 represents a haloalkyl group or the like, R 3 represents a hydrogen atom or the like, R 4 represents a haloalkyl group or the like, R 5 represents an alkyl group or the like, and m represents 0 or 2} or a salt thereof; an agricultural and horticultural insecticide comprising the compound or a salt thereof as an active ingredient; and a method for using the insecticide.
 (From EP2975039 A1)
机翻摘要
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地址
代理人
代理机构
优先权号
2013JP-0053201 2013JP-0107592 2013JP-0155074 2013JP-0231582 2014WO-JP56832
主权利要求
(BR112015020972)
1. Condensed heterocyclic, characterized by the general formula (1): (in which R 1 represents (1) an alkyl group (C 1-C 6);
 (2) an cyclcycle group (C 3-C 6);
 (3) a alcenil group (C 2-C 6);
 (4) an alcinil group (C 2-C 6);
 (5) a halo alkyl group (C 1-C 6);
 (6) a halogenalquil group (C 3-C 6);
 (7) a tar halo group (C 2-C 6);
 (8) a halo alcinil group (C 2-C 6);
 (9) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
 (10) a halo alcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
 (11) an cyclcycle group (C 3 -c 6) alkyl (C 1-C 6);
 (12) a halo cyclalalkyil group (C 3 -c 6) alkyl (C 1-C 6);
 (13) an albcoxi group (C 1 -c 6) halo alkyl (C 1-C 6);
 (14) a halo alkali group (C 1 -c 6) halo alkyl (C 1 -c 6);
 (15) an alkm group (C 1 -c 6) alkyl (C 1-C 6);
 (16) an alkylsulyl group (C 1 -c 6) alkyl (C 1 -c 6);
 (17) alkysulfonil (C 1 -c 6) alkyl (C 1 -c 6);
 (18) an alkyl group (C 1-C 6);
 (19) an alcoholic beverage group (C 1 -c 6) alkyl (C 1 -c 6);
 (20) an alkyamine group (C 1 -c 6) alkyl (C 1 -c 6) (where the alkyl groups of the alkylamino portion (C 1-C 6) may be equal or different);
 (21) a fenyl alquil group (C 1-C 6); or (22) a fenyl alquil group (C 1 -c 6) having, in the ring, 1 to 5 replacement groups selected from the group consisting of a halogen atom, (b) a group of halogens, (c) a group of alkyl groups (c) an alkyl group (C) an alkyl group (C 1 -c 6); (C 1-C 6), a halo alkyl group (C 1 -c 6) and (g) a halo alcoxi group (C 1 -c 6),
 R 2 represents (b 1) an halogen atom;
 (b) a cyane group;
 (b) a nitro group;
 (b) an alkyl group (C 1-C 6);
 (b) an cyclcycle group (C 3-C 6);
 (b) a alcenil group (C 2-C 6);
 (b) an alcinil group (C 2-C 6);
 (b) a halo alkyl group (C 1-C 6);
 (b) a halo cyclalalkyil group (C 3-C 6);
 (b) a tar halo group (C 2-C 6);
 (b) a halo alcinil group (C 2-C 6);
 (b) a group alkiliata (C 1-C 6);
 (b) an alkylsulyl group (C 1-C 6);
 (b) an alkilsulfonil group (C 1-C 6);
 (b) a halo alquilt group (C 1-C 6);
 (b 16) halo alkilsulyl (C 1 -c 6);
 (b) halo alkilsulfonil (C 1-C 6);
 (b) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
 (b) halo alcoxi (C 1 -c 6) alkyl (C 1 -c 6);
 (b) an cyclcycle group (C 3 -c 6) alkyl (C 1 -c 6);
 (b) a halo cyclalalkyil group (C 3 -c 6) alkyl (C 1 -c 6);
 (b) an albcoxi group (C 1 -c 6) halo alkyl (C 1 -c 6);
 (b) halo alkali alkyl (C 1 -c 6) halo alkyl (C 1 -c 6);
 (b) a hydrogen atom;
 (b) an albcoxi group (C 1 -c 6);
 (b) a halo alcoxi group (C 1 -c 6);
 (b) a friendly group;
 (b) an alkilamine group (C 1-C 6);
 (b) a di-alkilamino group (C 1-C 6) (in which the alkyl groups of the di alquil- (C 1-C 6) portion may be equal or different);
 (b) an alkylylamino group (C 1-C 6);
 (b) a group alkilsulphylamino (C 1-C 6);
 (b) an alkylsulphil group (C 1 -c 6) (amino (C 1 -c 6));
 (b) an alcoholic beverage group (C 1-C 6); or (b 34) a tri-alkilsilyl (C 1 -c 6) group (C 2 -c 6) (where the alkyl groups of tri-alkksilyl (C 1-C 6) can be equal or different),
 R 3 represents a hydrogen atom;
 R 4 represents (d 1) a hydrogen atom;
 (d) a halogen atom;
 (d) a cyane group;
 (d) a nitro group;
 (d) an alkyl group (C 1-C 6);
 (d) an albcoxi group (C 1 -c 6);
 (d) a group tragically (C 2-C 6);
 (d) an alcinilili group (C 2-C 6);
 (d) a halo alkyl group (C 1-C 6);
 (d) a halo alcoxi group (C 1 -c 6);
 (d) a halo tar group (C 2-C 6);
 (d) an alciniltoxic group (C 2-C 6);
 (d) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
 (d) halo alcoxi (C 1 -c 6) alkyl (C 1 -c 6);
 (d) an cyclcycle group (C 3 -c 6) alkyl (C 1 -c 6);
 (d) a halo cyclalalkyil group (C 3 -c 6) alkyl (C 1 -c 6);
 (d) an albcoxi group (C 1 -c 6) halo alkyl (C 1 -c 6);
 (d) a halo alkali group (C 1 -c 6) halo alkyl (C 1 -c 6);
 (d) a merchant group;
 (d) an alkiliata group (C 1-C 6);
 (d) an alkilcarbonilie group (C 1-C 6);
 (d) a halo alquilt group (C 1-C 6);
 (d) a fenil group;
 (d) a fenyl group having, in the ring, 1 to 5 replacement groups selected from the group consisting of (a) an halogen atom, (b) a cym group, (c) an alkyl group (c) an alkyl group (C 1 -c 6), (e) an albcoxi group (C 1 -c 6), a halo alkyl group (C 1 -c 6) and (g) a halo alcoxi group (C 1 C 6);
 (d) an alkylsulyl group (C 1-C 6);
 (d) an alkilsulfonil group (C 1-C 6);
 (d) halo alkilsulyl (C 1 -c 6); (d) a halo alkilsulfonil group (C 1-C 6),
 R 5 represents (and 1) a hydrogen atom;
 (and 2) a formil group;
 (and 3) an alkyl group (C 1-C 6);
 (and 4) an cyclcycle group (C 3-C 6);
 (5) a halo alkyl group (C 1-C 6);
 (6) a halo cyclalalkyil group (C 3-C 6);
 (and 7) an alkilsulfonil group (C 1-C 6);
 (and 8) halo alkilsulfonil (C 1-C 6);
 (and 9) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
 (10) a halo alcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
 (and 11) an albcoxi group (C 1 -c 6) halo alkyl (C 1 -c 6);
 (12) a halo alkali group (C 1 -c 6) halo alkyl (C 1 -c 6);
 (and 13) a friendly group; or (14) an albcoxi group (C 1-C 6),
 A and A 2 are, each, CH and A 3 is CH or N 0, 1, 2 or}, and a salt thereof.
2. Condensed heterocyclic, according to the claim that R 1 is (1) an alkyl group (C 1-C 6);
(2) an cyclcycle group (C 3-C 6);
(3) a alcenil group (C 2-C 6);
(4) an alcinil group (C 2-C 6);
(5) a halo alkyl group (C 1-C 6); (9) an albcoxi group (C 1-C 6) alkyl (C 1-C 6); (11) an cyclcycle group (C 3 -c 6) alkyl (C 1-C 6);
(15) alkyno group (C 1-C 6) alkyl (C 1-C 6);
(16) an alkylsulyl group (C 1 -c 6) alkyl (C 1 -c 6);
(17) alkysulfonil (C 1-C 6) alkyl (C 1-C 6);
(18) an alkyl group (C 1-C 6);
(19) an alcoholic beverage group (C 1 -c 6) alkyl (C 1 -c 6);
(20) an alkyamine group (C 1-C 6) alkyl (C 1-C 6) (where the alkyl groups of the alkylamino portion (C 1-C 6) may be equal or different);
(21) a fenyl alquil group (C 1-C 6); or (22) a fenyl alquil group (C 1 -c 6) having, in the ring, 1 to 5 replacement groups selected from the group consisting of a halogen atom, (b) a group of halogens, (c) a group of alkyl groups (c) an alkyl group (C) an alkyl group (C 1 -c 6); (C 1-C 6), a halo alkyl group (C 1 -c 6) and (g) a halo alcoxi group (C 1-C 6),
R 2 is (b 1) an halogen atom;
(b) an alkyl group (C 1-C 6);
(b) an cyclcycle group (C 3-C 6);
(b) a alcenil group (C 2-C 6);
(b) an alcinil group (C 2-C 6);
(b) a halo alkyl group (C 1-C 6); (b) a group alkiliata (C 1-C 6);
(b) a halo alquilt group (C 1-C 6);
(b 16) halo alkilsulyl (C 1 -c 6);
(b) halo alkilsulfonil (C 1-C 6);
(b) a hydrogen atom;
(b) an albcoxi group (C 1 -c 6);
(b) a halo alcoxi group (C 1 -c 6);
(b) a friendly group;
(b) a di-alkilamino group (C 1-C 6) (in which the alkyl groups of the di alquil- (C 1-C 6) portion may be equal or different);
(b) an alkylylamino group (C 1-C 6);
(b) a group alkilsulphylamino (C 1-C 6);
(b) an alkylsulphil group (C 1 -c 6) (amino (C 1 -c 6));
(b) an alcoholic beverage group (C 1-C 6); (b) a tri-alkilyl group (C 1 -c 6) alcinil (C 2 -c 6) (where the alkyyl groups of the tri-alkksilyl (C 1-C 6) portion may be equal or different),
R 3 is (c 1) a hydrogen atom,
R 4 is (d 2) an halogen atom; (d) an alkyl group (C 1-C 6); (d) a halo alkyl group (C 1-C 6);
(d) a merchant group;
(d) an alkiliata group (C 1-C 6);
(d) an alkilcarbonilie group (C 1-C 6);
(d) a halo alquilt group (C 1-C 6);
(d) a fenyl group having, in the ring, 1 to 5 replacement groups selected from the group consisting of (a) an halogen atom, (b) a cyrine group, (c) an alkyl group (c) an alkyl group (C 1-C 6), (e) an albcoxi group (C 1-C 6), a halo alkyl group (C 1-C 6) and (g) a halo alcoxi group (C 1-C 6), or (d 26) an alkylsulphil group (C 1-C 6),
R 5 is (and 3) an alkyl group (C 1-C 6);
(and 4) an cyclcycle group (C 3-C 6);
(5) a halo alkyl group (C 1-C 6); (and 9) an albcoxi group (C 1-C 6) alkyl (C 1-C 6);
(and 13) a friendly group; or (14) an albcoxi group (C 1 -c 6) and A and A 2 are each CH and A 3 is CH or A and a salt thereof.
3. Condensed heterocyclic, according to the claim that R 1 is (1) an alkyl group (C 1-C 6);
(2) an cyclcycle group (C 3-C 6);
(3) a alcenil group (C 2-C 6); (5) a halo alkyl group (C 1-C 6); (11) an cyclcycle group (C 3 -c 6) alkyl (C 1-C 6); (15) alkyno group (C 1-C 6) alkyl (C 1-C 6);
(18) an alkyl group (C 1-C 6);
(19) an alcoholic beverage group (C 1-C 6) alkyl (C 1-C 6);
(20) an alkyamine group (C 1 -c 6) alkyl (C 1 -c 6) (where the alkyl groups of the alkylamino portion (C 1-C 6) may be equal or different); or (22) a fenyl alkyl group (C 1-C 6) having, in the ring, 1 to 5 replacement groups selected from the group consisting of a halogen atom, (b) a group of halogens, (c) an alkyl group, (c) an alkyl group (C 1-C 6), an albcoxi group; (C 1-C 6), a halo alkyl group (C 1 -c 6) and (g) a halo alcoxi group (C 1 -c 6),
R 2 is (b 1) an halogen atom;
(b) an alkyl group (C 1-C 6);
(b) an cyclcycle group (C 3-C 6);
(b) a alcenil group (C 2-C 6);
(b) an alcinil group (C 2-C 6);
(b) a halo alkyl group (C 1-C 6); (b) a group alkiliata (C 1-C 6); (b) a halo alquilt group (C 1-C 6); (b) a hydrogen atom;
(b) a halo alcoxi group (C 1 -c 6);
(b) a friendly group;
(b) a di-alkilamino group (C 1-C 6) (in which the alkyl groups of the di alquil- (C 1-C 6) portion may be equal or different);
(b) an alkylylamino group (C 1-C 6);
(b) a group alkilsulphylamino (C 1-C 6);
(b) an alkylsulphil group (C 1 -c 6) (amino (C 1 -c 6));
(b) an alcoholic beverage group (C 1-C 6); (b) a tri-alkilyl group (C 1 -c 6) alcinil (C 2 -c 6) (where the alkyyl groups of the tri-alkksilyl (C 1-C 6) portion may be equal or different),
R 3 is (c 1) a hydrogen atom,
R 4 is (d 2) an halogen atom; (d) a halo alkyl group (C 1-C 6);
(d) a merchant group;
(d) an alkiliata group (C 1-C 6);
(d) an alkilcarbonilie group (C 1-C 6);
(d) a fenyl group having, in the ring, 1 to 5 replacement groups selected from the group consisting of (a) an halogen atom, (b) a cyrine group, (c) an alkyl group (c) an alkyl group (C 1-C 6), (e) an albcoxi group (C 1-C 6), a halo alkyl group (C 1-C 6) and (g) a halo alcoxi group (C 1-C 6); or (d 26) an alkilsulfonil group (C 1-C 6),
R 5 is (and 3) an alkyl group (C 1-C 6);
(and 4) an cyclcycle group (C 3-C 6); or (9) an albcoxi group (C 1 -c 6) alquil (C 1 -c 6), A 2 and A 3 are each CH and A is CH or N and a salt thereof.
4. Use of condensed heterocyclic composite compounds or a salt, as defined in any claim from 1 to 3, characterised by the fact that it is in the manufacture of an agricultural and horticultural insecticide.
5. Method of using an agricultural and horticulture insecticide, characterised by the fact that it understands to treat plants or soil with an active ingredient of the agricultural insecticide and horticulture according to the claim 4.
6. Method of controlling pests of agricultural and horticultural insects, characterised by the fact that it understands how to treat plants or soil with an effective quantity of agricultural and horticultural insecticide according to demand 4.
7. Disease control agent, characterised by the fact that it comprises condensed heterocyclic composite composite or a salt of it according to any of the claims 1 to 3 as an active ingredient.
8. Insecticide, characterised by the fact that it comprises a condensed heterocyclical compound containing imidazopiridazine or a salt from it according to any of the claims 1 to 3 as an active ingredient.
9. Condensed heterocyclic, characterized by the general formula (1):
in accordance with any of the claims from 1 to 3 in which R 1 represents (1) an alkyl group (C 1-C 6);
(2) an cyclcycle group (C 3-C 6);
(3) a alcenil group (C 2-C 6);
(4) an alcinil group (C 2-C 6);
(5) a halo alkyl group (C 1-C 6);
(6) a halogenalquil group (C 3-C 6);
(7) a tar halo group (C 2-C 6);
(8) a halo alcinil group (C 2-C 6);
(9) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
(10) a halo alcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
(11) an cyclcycle group (C 3 -c 6) alkyl (C 1-C 6);
(12) a halo cyclalalkyil group (C 3 -c 6) alkyl (C 1-C 6);
(13) an albcoxi group (C 1 -c 6) halo alkyl (C 1-C 6); (14) a halo alkali group (C 1 -c 6) halo alkyl (C 1 -c 6),
R 2 represents (b 1) an halogen atom;
(b) a cyane group;
(b) a nitro group;
(b) an alkyl group (C 1-C 6);
(b) a alcenil group (C 2-C 6);
(b) an alcinil group (C 2-C 6);
(b) a halo alkyl group (C 1-C 6);
(b) a halo cyclalalkyil group (C 3-C 6);
(b) a tar halo group (C 2-C 6);
(b) a halo alcinil group (C 2-C 6);
(b) a group alkiliata (C 1-C 6);
(b) an alkylsulyl group (C 1-C 6);
(b) an alkilsulfonil group (C 1-C 6);
(b) a halo alquilt group (C 1-C 6);
(b 16) halo alkilsulyl (C 1 -c 6);
(b) halo alkilsulfonil (C 1-C 6);
(b) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
(b) halo alcoxi (C 1 -c 6) alkyl (C 1 -c 6);
(b) an cyclcycle group (C 3 -c 6) alkyl (C 1 -c 6);
(b) a halo cyclalalkyil group (C 3 -c 6) alkyl (C 1 -c 6);
(b) an albcoxi group (C 1 -c 6) halo alkyl (C 1 -c 6); (b) a halo alkali group (C 1 -c 6) halo alkyl (C 1 -c 6),
R 3 represents (c 1) a hydrogen atom;
R 4 represents (d 1) a hydrogen atom;
(d) a halogen atom;
(d) a cyane group;
(d) a nitro group;
(d) an alkyl group (C 1-C 6);
(d) an albcoxi group (C 1 -c 6);
(d) a group tragically (C 2-C 6);
(d) an alcinilili group (C 2-C 6);
(d) a halo alkyl group (C 1-C 6);
(d) a halo alcoxi group (C 1 -c 6);
(d) a halo tar group (C 2-C 6);
(d) an alciniltoxic group (C 2-C 6);
(d) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
(d) halo alcoxi (C 1 -c 6) alkyl (C 1 -c 6);
(d) an cyclcycle group (C 3 -c 6) alkyl (C 1 -c 6);
(d) a halo cyclalalkyil group (C 3 -c 6) alkyl (C 1 -c 6);
(d) an albcoxi group (C 1 -c 6) halo alkyl (C 1 -c 6); or (d 18) a halo alkali group (C 1 -c 6) halo alquil (C 1 -c 6), R 5 represents (and 1) a hydrogen atom;
(and 2) a formil group;
(and 3) an alkyl group (C 1-C 6);
(and 4) an cyclcycle group (C 3-C 6);
(5) a halo alkyl group (C 1-C 6);
(6) a halo cyclalalkyil group (C 3-C 6);
(and 7) an alkilsulfonil group (C 1-C 6);
(and 8) halo alkilsulfonil (C 1-C 6);
(and 9) an albcoxi group (C 1 -c 6) alkyl (C 1 -c 6);
(10) a halo alcoxi group (C 1 -c 6) alkyl (C 1 -c 6); (1) an albcoxi group (C 1 -c 6) halo alkyl (C 1-C 6); or (12) a halo alkali group (C 1 -c 6) halo alkyl (C 1 -c 6), A and A 2 are CH, A 3, CH and A 0 is CH or N 2, and a salt of it.
法律状态
GRANTED
专利类型码
B1 A2 A1
国别省市代码
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